PDB クエリの検索結果 - 日本蛋白質構造データバンク

PDB: 1 件

Structure of CDK12/CycK in complex with a small molecule inhibitor N-(4-(1-methyl-1H-pyrazol-4-yl)phenyl)-N-((1r,4r)-4-(quinazolin-2-ylamino)cyclohexyl)acetamide
分子名称:	Cyclin-K, Cyclin-dependent kinase 12, MAGNESIUM ION, ...
著者	Klein, M.G.
登録日	2018-03-01
公開日	2018-08-29
最終更新日	2018-09-26
実験手法	X-RAY DIFFRACTION (2.8 Å)
主引用文献	Discovery of 3-Benzyl-1-( trans-4-((5-cyanopyridin-2-yl)amino)cyclohexyl)-1-arylurea Derivatives as Novel and Selective Cyclin-Dependent Kinase 12 (CDK12) Inhibitors. J. Med. Chem., 61, 2018