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PDB: 1 件

6BQ0
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BU of 6bq0 by Molmil
Structure of human monoacylglycerol lipase bound to a covalent inhibitor
分子名称: 1-({(1R,5S,6r)-6-[1-(4-fluorophenyl)-1H-pyrazol-3-yl]-3-azabicyclo[3.1.0]hexane-3-carbonyl}oxy)pyrrolidine-2,5-dione, Monoglyceride lipase
著者Pandit, J.
登録日2017-11-27
公開日2018-03-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation.
J. Med. Chem., 61, 2018

221051

件を2024-06-12に公開中

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