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PDB: 2 件

9DCD
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BU of 9dcd by Molmil
Structure of J-PKAc chimera in complex with Aplithianine d2
分子名称: N-(2-aminoethyl)-4-(7H-purin-6-yl)-3,4-dihydro-2H-1,4-thiazine-6-carboxamide, cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha
著者Martinez Fiesco, J.A, Zhang, P.
登録日2024-08-25
公開日2025-07-09
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Chemical Evolution of Aplithianine Class of Serine/Threonine Kinase Inhibitors.
J.Med.Chem., 68, 2025
9DC6
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BU of 9dc6 by Molmil
Structure of J-PKAc chimera in complex with Aplithianine e1
分子名称: N-(2-aminoethyl)-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-3,4-dihydro-2H-1,4-thiazine-6-carboxamide, cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha
著者Martinez Fiesco, J.A, Zhang, P.
登録日2024-08-25
公開日2025-07-09
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Chemical Evolution of Aplithianine Class of Serine/Threonine Kinase Inhibitors.
J.Med.Chem., 68, 2025

238582

件を2025-07-09に公開中

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