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PDB: 1 件

8V42
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Structure of Human Vaccinia-related Kinase 1 (VRK1) Bound to ACH000400
分子名称: (7S)-2-(3,5-difluoro-4-hydroxyanilino)-7-methyl-5-[(1,2-oxazol-5-yl)methyl]-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5H)-one, DI(HYDROXYETHYL)ETHER, SULFATE ION, ...
著者Counago, R.M, de Souza, G.P, Azevedo, A, Guimaraes, C, Mascarello, A, Gama, F, Ferreira, M, Arruda, P.
登録日2023-11-28
公開日2024-09-04
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Novel Dihydropteridinone Derivatives As Potent Inhibitors of the Understudied Human Kinases Vaccinia-Related Kinase 1 and Casein Kinase 1 delta / epsilon.
J.Med.Chem., 67, 2024

225681

件を2024-10-02に公開中

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