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PDB: 1 件

8K5R
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CDK9/cyclin T1 in complex with KB-0742
分子名称: (1S,3S)-N3-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamine, Cyclin-T1, Cyclin-dependent kinase 9
著者Zhou, M, Li, H, Gao, H, Trotter, B.W, Freeman, D.
登録日2023-07-24
公開日2023-12-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (3.751 Å)
主引用文献Discovery of KB-0742, a Potent, Selective, Orally Bioavailable Small Molecule Inhibitor of CDK9 for MYC-Dependent Cancers.
J.Med.Chem., 66, 2023

222036

件を2024-07-03に公開中

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