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PDB: 3 件

7PJR
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BU of 7pjr by Molmil
Notum_ARUK3000438
分子名称: 1-[4-chloranyl-3-(trifluoromethyl)phenyl]-1,2,3-triazole, 2-acetamido-2-deoxy-beta-D-glucopyranose, DIMETHYL SULFOXIDE, ...
著者Vecchia, L, Zhao, Y, Fish, P, Jones, E.Y.
登録日2021-08-24
公開日2022-09-07
最終更新日2023-03-22
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit.
J.Med.Chem., 65, 2022
7PK3
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BU of 7pk3 by Molmil
Notum_ARUK3001185
分子名称: 1-[2,4-bis(chloranyl)-3-(trifluoromethyl)phenyl]-1,2,3-triazole, 2-acetamido-2-deoxy-beta-D-glucopyranose, DIMETHYL SULFOXIDE, ...
著者Vecchia, L, Hillier, J, Zhao, Y, Fish, P, Jones, E.Y.
登録日2021-08-25
公開日2022-09-07
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.41 Å)
主引用文献Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit.
J.Med.Chem., 65, 2022
7PKV
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BU of 7pkv by Molmil
Notum_Inhibitor ARUK3000223
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, DIMETHYL SULFOXIDE, Palmitoleoyl-protein carboxylesterase NOTUM, ...
著者Ruza, R, Zhao, Y, Fish, P, Jones, E.Y.
登録日2021-08-26
公開日2022-09-07
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit.
J.Med.Chem., 65, 2022

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件を2024-07-10に公開中

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