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PDB: 1 件

Crystal structure of BRD4(1) bound to the dual BET-HDAC inhibitor LSH24
分子名称:	4-acetyl-3-ethyl-N-(3-(3-(hydroxyamino)-3-oxopropyl)phenyl)-5-methyl-1H-pyrrole-2-carboxamide, Bromodomain-containing protein 4
著者	Huegle, M.
登録日	2020-11-10
公開日	2021-10-06
最終更新日	2024-01-31
実験手法	X-RAY DIFFRACTION (1.5 Å)
主引用文献	4-Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for Hybrid Inhibitors of BET Proteins and Histone Deacetylases as Antileukemia Drug Leads. J.Med.Chem., 64, 2021