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PDB: 1 件

7F0I
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phosphodiesterase-9A in complex with inhibitor 4b
分子名称: 1-cyclopentyl-6-[[(2R)-1-(6-fluoranyl-2-azaspiro[3.3]heptan-2-yl)-1-oxidanylidene-propan-2-yl]amino]-5H-pyrazolo[3,4-d]pyrimidin-4-one, Isoform PDE9A2 of High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A, MAGNESIUM ION, ...
著者Wu, Y, Huang, Y.Y, Luo, H.B.
登録日2021-06-04
公開日2022-04-13
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.70000887 Å)
主引用文献Discovery of Potent Phosphodiesterase-9 Inhibitors for the Treatment of Hepatic Fibrosis
J.Med.Chem., 64, 2021

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件を2024-09-11に公開中

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