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PDB: 1 件

7N7X
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Crystal structure of BCX7353(ORLADEYO) in complex with human plasma kallikrein serine protease domain at 2.1 angstrom resolution
分子名称: Orladeyo, PHOSPHATE ION, Plasma kallikrein light chain
著者Krishnan, R, Yarlagadda, B.S, Kotian, P, Polach, K.J, Zhang, W.
登録日2021-06-11
公開日2021-09-15
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.097 Å)
主引用文献Berotralstat (BCX7353): Structure-Guided Design of a Potent, Selective, and Oral Plasma Kallikrein Inhibitor to Prevent Attacks of Hereditary Angioedema (HAE).
J.Med.Chem., 64, 2021

238582

件を2025-07-09に公開中

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