PDB クエリの検索結果 - 日本蛋白質構造データバンク

PDB: 2 件

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 with GSK789
分子名称:	(3~{R},4~{R})-~{N}-cyclohexyl-4-[[5-(furan-2-yl)-3-methyl-2-oxidanylidene-1~{H}-1,7-naphthyridin-8-yl]amino]-1-methyl-piperidine-3-carboxamide, Bromodomain-containing protein 4
著者	Chung, C.
登録日	2020-05-31
公開日	2020-07-29
最終更新日	2024-05-01
実験手法	X-RAY DIFFRACTION (1.624 Å)
主引用文献	GSK789: A Selective Inhibitor of the First Bromodomains (BD1) of the Bromo and Extra Terminal Domain (BET) Proteins. J.Med.Chem., 63, 2020

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 (3R,4R)-N-cyclohexyl-4-((3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)piperidine-3-carboxamide
分子名称:	(3R,4R)-N-cyclohexyl-4-((3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)piperidine-3-carboxamide, Bromodomain-containing protein 4
著者	Chung, C.
登録日	2020-05-31
公開日	2020-07-29
最終更新日	2024-05-01
実験手法	X-RAY DIFFRACTION (1.26 Å)
主引用文献	GSK789: A Selective Inhibitor of the First Bromodomains (BD1) of the Bromo and Extra Terminal Domain (BET) Proteins. J.Med.Chem., 63, 2020