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PDB: 1 件

8FE9
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Crystal structure of Ack1 kinase K161Q mutant in complex with the selective inhibitor (R)-9b
分子名称: 5-chloro-N~2~-[4-(4-methylpiperazin-1-yl)phenyl]-N~4~-{[(2R)-oxolan-2-yl]methyl}pyrimidine-2,4-diamine, Activated CDC42 kinase 1
著者Paung, Y, Kan, Y, Seeliger, M.S, Miller, W.T.
登録日2022-12-06
公開日2023-03-29
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Biochemical Studies of Systemic Lupus Erythematosus-Associated Mutations in Nonreceptor Tyrosine Kinases Ack1 and Brk.
Biochemistry, 62, 2023

238582

件を2025-07-09に公開中

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