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PDB: 1 件

9QB5
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AP2-associated protein kinase 1 (AAK1) bound to CKJB68
分子名称: AP2-associated protein kinase 1, SULFATE ION, ~{N}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide
著者Preuss, F, Mensing, T.E, Hanke, T, Knapp, S, Mathea, S.
登録日2025-02-28
公開日2025-04-09
最終更新日2025-10-22
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.
Eur.J.Med.Chem., 299, 2025

245396

件を2025-11-26に公開中

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