9KLB
 
 | | G9a in complex with RK-133232 (compound 16g) | | 分子名称: | Histone-lysine N-methyltransferase EHMT2, SINEFUNGIN, ZINC ION, ... | | 著者 | Niwa, H, Shirai, F, Sato, S, Nishigaya, Y, Ihara, K, Shirouzu, M, Umehara, T. | | 登録日 | 2024-11-14 | | 公開日 | 2025-05-21 | | 最終更新日 | 2025-06-04 | | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | | 主引用文献 | Discovery of potent substrate-type lysine methyltransferase G9a inhibitors for the treatment of sickle cell disease.
Eur.J.Med.Chem., 293, 2025
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9KLC
 | | G9a in complex with the S-isomer of RK-131902 (racemic compound rac-10a) | | 分子名称: | Histone-lysine N-methyltransferase EHMT2, SINEFUNGIN, ZINC ION, ... | | 著者 | Niwa, H, Shirai, F, Sato, S, Nishigaya, Y, Ihara, K, Shirouzu, M, Umehara, T. | | 登録日 | 2024-11-14 | | 公開日 | 2025-05-21 | | 最終更新日 | 2025-06-04 | | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | | 主引用文献 | Discovery of potent substrate-type lysine methyltransferase G9a inhibitors for the treatment of sickle cell disease.
Eur.J.Med.Chem., 293, 2025
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