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PDB: 1 件

5NJH
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Triazolopyrimidines stabilize microtubules by binding to the vinca inhibitor site of tubulin
分子名称: 5-chloranyl-7-[(1~{R},5~{S})-3-methoxy-8-azabicyclo[3.2.1]octan-8-yl]-6-[2,4,6-tris(fluoranyl)phenyl]-[1,2,4]triazolo[1,5-a]pyrimidine, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Sharma, A, Calvo, G.S, Prota, A.E, Diaz, J.F, Steinmetz, M.O.
登録日2017-03-28
公開日2017-06-21
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.394 Å)
主引用文献Triazolopyrimidines Are Microtubule-Stabilizing Agents that Bind the Vinca Inhibitor Site of Tubulin.
Cell Chem Biol, 24, 2017

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件を2024-07-24に公開中

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