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PDB: 1 件

2R0U
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Crystal Structure of Chek1 in Complex with Inhibitor 54
分子名称: 6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1H-pyrazol-4-yl)benzo[h]isoquinolin-1(2H)-one, Serine/threonine-protein kinase Chk1
著者Yan, Y, Ikuta, M.
登録日2007-08-21
公開日2007-10-30
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Synthesis and evaluation of substituted benzoisoquinolinones as potent inhibitors of Chk1 kinase.
Bioorg.Med.Chem.Lett., 17, 2007

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件を2024-07-24に公開中

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