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PDB: 1 件

4JZR
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Structure of Prolyl Hydroxylase Domain-containing Protein (PHD) with Inhibitors
分子名称: 1,2-ETHANEDIOL, 2-(biphenyl-4-yl)-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-1-one, Egl nine homolog 1, ...
著者Ma, Y, Yang, L.
登録日2013-04-03
公開日2013-10-30
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Novel complex crystal structure of prolyl hydroxylase domain-containing protein 2 (PHD2): 2,8-Diazaspiro[4.5]decan-1-ones as potent, orally bioavailable PHD2 inhibitors
Bioorg.Med.Chem., 21, 2013

222624

件を2024-07-17に公開中

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