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PDB: 3 件

8IMF
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BU of 8imf by Molmil
Human cGAS catalytic domain bound with baicalein
分子名称: 5,6,7-trihydroxy-2-phenyl-4H-chromen-4-one, Cyclic GMP-AMP synthase, ZINC ION
著者Zhao, W.F, Xu, Y.C.
登録日2023-03-06
公開日2024-01-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Discovery of novel cGAS inhibitors based on natural flavonoids.
Bioorg.Chem., 140, 2023
8IME
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BU of 8ime by Molmil
Human cGAS catalytic domain bound with baicalin
分子名称: 5,6-dihydroxy-4-oxo-2-phenyl-4H-chromen-7-yl beta-D-glucopyranosiduronic acid, Cyclic GMP-AMP synthase, ZINC ION
著者Zhao, W.F, Xu, Y.C.
登録日2023-03-06
公開日2024-01-03
実験手法X-RAY DIFFRACTION (2.63 Å)
主引用文献Discovery of novel cGAS inhibitors based on natural flavonoids.
Bioorg.Chem., 140, 2023
8IMG
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BU of 8img by Molmil
Human cGAS catalytic domain bound with C20
分子名称: 2-[2-hydroxy-2-oxoethyl-[3-(7-methoxy-4-methyl-2-oxidanylidene-chromen-3-yl)propanoyl]amino]ethanoic acid, Cyclic GMP-AMP synthase, ZINC ION
著者Zhao, W.F, Li, J.M, Xu, Y.C.
登録日2023-03-06
公開日2024-01-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Discovery of novel cGAS inhibitors based on natural flavonoids.
Bioorg.Chem., 140, 2023

222415

件を2024-07-10に公開中

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