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PDB: 2 件

5DW1
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BU of 5dw1 by Molmil
X-ray crystal structure of human BRD2(BD2) in complex with RVX297 to 1.55 A resolution
分子名称: 2-{3,5-dimethyl-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-5,7-dimethoxyquinazolin-4(3H)-one, Bromodomain-containing protein 2, SODIUM ION
著者White, A, Fontano, E, Suto, R.K.
登録日2015-09-22
公開日2016-06-22
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献RVX-297- a novel BD2 selective inhibitor of BET bromodomains.
Biochem.Biophys.Res.Commun., 477, 2016
5DW2
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BU of 5dw2 by Molmil
X-ray crystal structure of human BRD4(BD1) in complex with RVX297 to 1.12 A resolution
分子名称: 1,2-ETHANEDIOL, 2-{3,5-dimethyl-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-5,7-dimethoxyquinazolin-4(3H)-one, Bromodomain-containing protein 4
著者White, A, Fontano, E, Suto, R.K.
登録日2015-09-22
公開日2016-06-22
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.12 Å)
主引用文献RVX-297- a novel BD2 selective inhibitor of BET bromodomains.
Biochem.Biophys.Res.Commun., 477, 2016

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件を2024-08-07に公開中

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