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PDB: 1 件

8P8C
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HUMAN CD38 ECTODOMAIN BOUND TO COMPOUND 9-ADPR ADDUCT
分子名称: ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1, [[(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methoxy-oxidanyl-phosphoryl] [(2~{R},3~{S},4~{R},5~{R})-5-[4-[4-[[4-(2-methoxyethoxy)cyclohexyl]amino]-1-methyl-2-oxidanylidene-quinolin-6-yl]pyrazol-1-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl hydrogen phosphate
著者Rangel, V, Zebisch, M, Doyle, K.J, Burli, R.W.
登録日2023-05-31
公開日2023-07-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.653 Å)
主引用文献A Covalent Binding Mode of a Pyrazole-Based CD38 Inhibitor
Helv.Chim.Acta, 106, 2023

222415

件を2024-07-10に公開中

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