9BAJ
 
 | Crystal structure of GDP-bound human K-RAS in a covalent complex with aryl sulfonyl fluoride compounds. | 分子名称: | 3-(dioxo-lambda~6~-sulfanyl)-N-phenylbenzene-1-sulfonamide, GUANOSINE-5'-DIPHOSPHATE, Isoform 2B of GTPase KRas, ... | 著者 | Landgraf, A.D, Brenner, R.J, Ghozayel, M.K, Bum-Erdene, K, Gonzalez-Gutierrez, G, Meroueh, S. | 登録日 | 2024-04-04 | 公開日 | 2025-04-09 | 最終更新日 | 2025-07-02 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | Small-Molecule KRAS Inhibitors by Tyrosine Covalent Bond Formation. Chemmedchem, 20, 2025
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9BAK
 
 | Crystal structure of GDP-bound human K-RAS in a covalent complex with aryl sulfonyl fluoride compounds. | 分子名称: | 3-[bis(oxidanylidene)-$l^{5}-sulfanyl]-~{N}-pyridazin-3-yl-benzenesulfonamide, GUANOSINE-5'-DIPHOSPHATE, Isoform 2B of GTPase KRas, ... | 著者 | Landgraf, A.D, Brenner, R.J, Ghozayel, M.K, Bum-Erdene, K, Gonzalez-Gutierrez, G, Meroueh, S. | 登録日 | 2024-04-04 | 公開日 | 2025-04-09 | 最終更新日 | 2025-07-02 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Small-Molecule KRAS Inhibitors by Tyrosine Covalent Bond Formation. Chemmedchem, 20, 2025
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9BAI
 
 | Crystal structure of GDP-bound human K-RAS in a covalent complex with aryl sulfonyl fluoride compounds. | 分子名称: | 3-[bis(oxidanylidene)-$l^{5}-sulfanyl]-~{N}-pyridin-4-yl-benzenesulfonamide, GUANOSINE-5'-DIPHOSPHATE, Isoform 2B of GTPase KRas, ... | 著者 | Landgraf, A.D, Brenner, R.J, Ghozayel, M.K, Bum-Erdene, K, Gonzalez-Gutierrez, G, Meroueh, S. | 登録日 | 2024-04-04 | 公開日 | 2025-04-09 | 最終更新日 | 2025-07-02 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | Small-Molecule KRAS Inhibitors by Tyrosine Covalent Bond Formation. Chemmedchem, 20, 2025
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