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PDB: 8 件

8FPQ
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BU of 8fpq by Molmil
PCSK9 in complex with an inhibitor
分子名称: CALCIUM ION, MCR-PHE-VAL-PRO-THR-THR-BIF-MAA-BIF-MAA-GLU-ALA-PRO-ALA-NEH inhibitor, Proprotein convertase subtilisin/kexin type 9
著者Xu, M, Chopra, R.
登録日2023-01-05
公開日2024-10-16
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (2.503 Å)
主引用文献Discovery of Truncated Cyclic Peptides Targeting an Induced-Fit Pocket on PCSK9.
Chemmedchem, 19, 2024
8FPO
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BU of 8fpo by Molmil
PCSK9 in complex with an inhibitor
分子名称: CALCIUM ION, MCR-ALA-7T2-GLY-004-7T2-SER-7T2-0NC inhibitor, Proprotein convertase subtilisin/kexin type 9
著者Xu, M, Chopra, R.
登録日2023-01-05
公開日2024-10-16
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (2.997 Å)
主引用文献Discovery of Truncated Cyclic Peptides Targeting an Induced-Fit Pocket on PCSK9.
Chemmedchem, 19, 2024
8FVO
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BU of 8fvo by Molmil
PCSK9 in complex with an inhibitor
分子名称: CALCIUM ION, MCR-ALA-7T2-GLY-004-7T2-SER-7T2-ALA-GLY-NH2 inhibitor, Proprotein convertase subtilisin/kexin type 9
著者Xu, M, Chopra, R.
登録日2023-01-19
公開日2024-10-16
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (2.652 Å)
主引用文献Discovery of Truncated Cyclic Peptides Targeting an Induced-Fit Pocket on PCSK9.
Chemmedchem, 19, 2024
8FVP
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BU of 8fvp by Molmil
PCSK9 in complex with an inhibitor
分子名称: CALCIUM ION, PPI-YD5-NLE-7T2-SER-7T2-DPP-GLY-NH2 inhibitor, Proprotein convertase subtilisin/kexin type 9
著者Xu, M, Chopra, R.
登録日2023-01-19
公開日2024-10-16
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (2.602 Å)
主引用文献Discovery of Truncated Cyclic Peptides Targeting an Induced-Fit Pocket on PCSK9.
Chemmedchem, 19, 2024
8FVQ
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BU of 8fvq by Molmil
PCSK9 in complex with an inhibitor
分子名称: ACE-PHE-VAL-DAB-THR-THR-PHE-MAA-BIF-YBR inhibitor, Proprotein convertase subtilisin/kexin type 9
著者Xu, M, Chopra, R.
登録日2023-01-19
公開日2024-10-16
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献Discovery of Truncated Cyclic Peptides Targeting an Induced-Fit Pocket on PCSK9.
Chemmedchem, 19, 2024
8FVL
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BU of 8fvl by Molmil
PCSK9 in complex with an inhibitor
分子名称: Proprotein convertase subtilisin/kexin type 9, YBX-YC3-VAL-PRO-THR-THR-PHE-MAA-CYS-MN1 inhibitor
著者Xu, M, Chopra, R.
登録日2023-01-19
公開日2024-10-16
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (1.961 Å)
主引用文献Discovery of Truncated Cyclic Peptides Targeting an Induced-Fit Pocket on PCSK9.
Chemmedchem, 19, 2024
8FVM
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BU of 8fvm by Molmil
PCSK9 in complex with an inhibitor
分子名称: CALCIUM ION, DGN-DVA-YC3-GLU-PRO-THR-THR-PHE-MAA-A1BC0 inhibitor, Proprotein convertase subtilisin/kexin type 9
著者Xu, M, Chopra, R.
登録日2023-01-19
公開日2024-10-16
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (2.852 Å)
主引用文献Discovery of Truncated Cyclic Peptides Targeting an Induced-Fit Pocket on PCSK9.
Chemmedchem, 19, 2024
8FVN
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BU of 8fvn by Molmil
PCSK9 in complex with an inhibitor
分子名称: MCR-ALO-MAA-ALA-MAA-NLE-7T2-SER-7T2-ALA-NH2 inhibitor, Proprotein convertase subtilisin/kexin type 9
著者Xu, M, Chopra, R.
登録日2023-01-19
公開日2024-10-16
最終更新日2025-04-30
実験手法X-RAY DIFFRACTION (2.71 Å)
主引用文献Discovery of Truncated Cyclic Peptides Targeting an Induced-Fit Pocket on PCSK9.
Chemmedchem, 19, 2024

238582

件を2025-07-09に公開中

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