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PDB: 1 件

5NGB
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X-Ray Diffraction Crystal Structure of the murine PI3K p110delta in complex with a pan inhibitor
分子名称: 3-[[4-(2-morpholin-4-yl-4-oxidanylidene-3~{H}-quinolin-8-yl)-1,2,3-triazol-1-yl]methyl]benzoic acid, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Berndt, A, Williams, R.L.
登録日2017-03-17
公開日2017-09-13
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs.
ChemMedChem, 12, 2017

222415

件を2024-07-10に公開中

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