PDB クエリの検索結果 - 日本蛋白質構造データバンク

PDB: 2 件

Crystal Structure of AKT1 in Complex with Covalent-Allosteric AKT Inhibitor 16a
分子名称:	RAC-alpha serine/threonine-protein kinase, ~{N}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{H}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{H}-benzimidazol-5-yl]propanamide
著者	Landel, I, Mueller, M.P, Rauh, D.
登録日	2019-07-15
公開日	2019-10-16
最終更新日	2024-01-24
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Covalent-Allosteric Inhibitors to Achieve Akt Isoform-Selectivity. Angew.Chem.Int.Ed.Engl., 58, 2019

Crystal Structure of AKT1 in Complex with Covalent-Allosteric AKT Inhibitor 15c
分子名称:	RAC-alpha serine/threonine-protein kinase, ~{N}-[3-[1-[[4-[5-[(4-hydroxyphenyl)methyl]-6-oxidanylidene-2-phenyl-1~{H}-pyrazin-3-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{H}-benzimidazol-5-yl]propanamide
著者	Landel, I, Mueller, M.P, Rauh, D.
登録日	2019-07-15
公開日	2019-10-16
最終更新日	2024-01-24
実験手法	X-RAY DIFFRACTION (2.6 Å)
主引用文献	Covalent-Allosteric Inhibitors to Achieve Akt Isoform-Selectivity. Angew.Chem.Int.Ed.Engl., 58, 2019