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PDB: 4 件

5MFP
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BU of 5mfp by Molmil
Human Sirt6 in complex with activator UBCS58
分子名称: 1,2-ETHANEDIOL, 4-pyridin-3-ylpyrrolo[1,2-a]quinoxaline, NAD-dependent protein deacetylase sirtuin-6, ...
著者Steegborn, C, You, W, Kambach, C.
登録日2016-11-18
公開日2016-12-28
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献Structural Basis of Sirtuin 6 Activation by Synthetic Small Molecules.
Angew. Chem. Int. Ed. Engl., 56, 2017
5MF6
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BU of 5mf6 by Molmil
Human Sirt6 in complex with activator UBCS039
分子名称: (4~{R})-4-pyridin-3-yl-4,5-dihydropyrrolo[1,2-a]quinoxaline, 1,2-ETHANEDIOL, NAD-dependent protein deacetylase sirtuin-6, ...
著者Steegborn, C, You, W, Kambach, C.
登録日2016-11-17
公開日2016-12-28
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Structural Basis of Sirtuin 6 Activation by Synthetic Small Molecules.
Angew. Chem. Int. Ed. Engl., 56, 2017
5MFZ
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BU of 5mfz by Molmil
Human Sirt6 in complex with small molecule UBCS40
分子名称: 1,2-ETHANEDIOL, 1-pyrrolo[1,2-a]quinoxalin-4-ylnaphthalen-2-ol, NAD-dependent protein deacetylase sirtuin-6, ...
著者Steegborn, C, You, W, Kambach, C.
登録日2016-11-19
公開日2016-12-28
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural Basis of Sirtuin 6 Activation by Synthetic Small Molecules.
Angew. Chem. Int. Ed. Engl., 56, 2017
5MGN
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BU of 5mgn by Molmil
Human Sirt6 in complex with activator UBCS38
分子名称: (4~{R})-4-pyridin-3-yl-5-[3-(trifluoromethyl)phenyl]sulfonyl-4~{H}-pyrrolo[1,2-a]quinoxaline, 1,2-ETHANEDIOL, NAD-dependent protein deacetylase sirtuin-6, ...
著者Steegborn, C, You, W, Kambach, C.
登録日2016-11-21
公開日2016-12-28
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Structural Basis of Sirtuin 6 Activation by Synthetic Small Molecules.
Angew. Chem. Int. Ed. Engl., 56, 2017

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件を2024-07-10に公開中

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