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PDB: 1 件

4DRU
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HCV NS5B in complex with macrocyclic INDOLE INHIBITOR
分子名称: 13-cyclohexyl-3-methoxy-17,22-dimethyl-7H-10,6-(methanoiminothioiminobutanoiminomethano)indolo[2,1-a][2]benzazepine-14,23-dione 16,16-dioxide, GLYCEROL, RNA-directed RNA polymerase, ...
著者Cummings, M.D, Vendeville, S.
登録日2012-02-17
公開日2012-04-18
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure-based macrocyclization yields hepatitis C virus NS5B inhibitors with improved binding affinities and pharmacokinetic properties.
Angew.Chem.Int.Ed.Engl., 51, 2012

222624

件を2024-07-17に公開中

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