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PDB: 3 results

5VED
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BU of 5ved by Molmil
PAK4 kinase domain in complex with Staurosporine
Descriptor: STAUROSPORINE, Serine/threonine-protein kinase PAK 4
Authors:Zhang, E.Y, Ha, B.H, Boggon, T.J.
Deposit date:2017-04-04
Release date:2017-10-18
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.301 Å)
Cite:PAK4 crystal structures suggest unusual kinase conformational movements.
Biochim. Biophys. Acta, 1866, 2018
5VEF
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BU of 5vef by Molmil
PAK4 kinase domain in complex with fasudil
Descriptor: 5-(1,4-DIAZEPAN-1-SULFONYL)ISOQUINOLINE, ACETATE ION, Serine/threonine-protein kinase PAK 4
Authors:Zhang, E.Y, Ha, B.H, Boggon, T.J.
Deposit date:2017-04-04
Release date:2017-10-18
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.752 Å)
Cite:PAK4 crystal structures suggest unusual kinase conformational movements.
Biochim. Biophys. Acta, 1866, 2018
5VEE
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BU of 5vee by Molmil
PAK4 kinase domain in complex with FRAX486
Descriptor: 6-(2,4-dichlorophenyl)-8-ethyl-2-{[3-fluoro-4-(piperazin-1-yl)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8H)-one, Serine/threonine-protein kinase PAK 4
Authors:Zhang, E.Y, Ha, B.H, Boggon, T.J.
Deposit date:2017-04-04
Release date:2017-10-18
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:PAK4 crystal structures suggest unusual kinase conformational movements.
Biochim. Biophys. Acta, 1866, 2018

222415

数据于2024-07-10公开中

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