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PDB: 6 件

3K2M
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BU of 3k2m by Molmil
Crystal Structure of Monobody HA4/Abl1 SH2 Domain Complex
分子名称: Monobody HA4, PHOSPHATE ION, Proto-oncogene tyrosine-protein kinase ABL1
著者Wojcik, J.B, Duguid, E.
登録日2009-09-30
公開日2010-03-31
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献A potent and highly specific FN3 monobody inhibitor of the Abl SH2 domain.
Nat.Struct.Mol.Biol., 17, 2010
3T04
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BU of 3t04 by Molmil
Crystal structure of monobody 7c12/abl1 sh2 domain complex
分子名称: GLYCEROL, MONOBODY 7C12, SULFATE ION, ...
著者Wojcik, J.B, Wyrzucki, A.M, Koide, S.
登録日2011-07-19
公開日2011-11-23
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Targeting the SH2-Kinase Interface in Bcr-Abl Inhibits Leukemogenesis.
Cell(Cambridge,Mass.), 147, 2011
3UYO
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Crystal structure of monobody SH13/ABL1 SH2 domain complex
分子名称: Monobody SH13, SULFATE ION, Tyrosine-protein kinase ABL1
著者Wojcik, J.B, Koide, A, Koide, S.
登録日2011-12-06
公開日2011-12-28
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献Teaching an old scaffold new tricks: monobodies constructed using alternative surfaces of the FN3 scaffold.
J.Mol.Biol., 415, 2012
5DC0
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BU of 5dc0 by Molmil
CRYSTAL STRUCTURE OF MONOBODY GG3/ABL1 SH2 DOMAIN COMPLEX
分子名称: Fibronectin, Tyrosine-protein kinase ABL1
著者Wojcik, J.B, Grabe, G, Koide, S.
登録日2015-08-22
公開日2016-03-02
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献Allosteric Inhibition of Bcr-Abl Kinase by High Affinity Monobody Inhibitors Directed to the Src Homology 2 (SH2)-Kinase Interface.
J.Biol.Chem., 291, 2016
5DC9
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BU of 5dc9 by Molmil
CRYSTAL STRUCTURE OF MONOBODY AS25/ABL1 SH2 DOMAIN COMPLEX, CRYSTAL B
分子名称: AS25 monobody, GLYCEROL, IMIDAZOLE, ...
著者Wojcik, J.B, Koide, A, Koide, S.
登録日2015-08-23
公開日2016-03-02
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Allosteric Inhibition of Bcr-Abl Kinase by High Affinity Monobody Inhibitors Directed to the Src Homology 2 (SH2)-Kinase Interface.
J.Biol.Chem., 291, 2016
5DC4
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BU of 5dc4 by Molmil
CRYSTAL STRUCTURE OF MONOBODY AS25/ABL1 SH2 DOMAIN COMPLEX, CRYSTAL A
分子名称: AS25 monobody, GLYCEROL, Tyrosine-protein kinase ABL1
著者Wojcik, J.B, Koide, A, Koide, S.
登録日2015-08-23
公開日2016-03-02
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.48 Å)
主引用文献Allosteric Inhibition of Bcr-Abl Kinase by High Affinity Monobody Inhibitors Directed to the Src Homology 2 (SH2)-Kinase Interface.
J.Biol.Chem., 291, 2016

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件を2024-08-07に公開中

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