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PDB: 7 件

1Y9O
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1H NMR Structure of Acylphosphatase from the hyperthermophile Sulfolobus Solfataricus
分子名称: Acylphosphatase
著者Corazza, A, Rosano, C, Pagano, K, Alverdi, V, Esposito, G, Capanni, C, Bemporad, F, Plakoutsi, G, Stefani, M, Chiti, F, Zuccotti, S, Bolognesi, M, Viglino, P.
登録日2004-12-16
公開日2005-11-29
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Structure, conformational stability, and enzymatic properties of acylphosphatase from the hyperthermophile Sulfolobus solfataricus
Proteins, 62, 2006
1PHR
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THE CRYSTAL STRUCTURE OF A LOW MOLECULAR PHOSPHOTYROSINE PROTEIN PHOSPHATASE
分子名称: LOW MOLECULAR WEIGHT PHOSPHOTYROSINE PROTEIN PHOSPHATASE, SULFATE ION
著者Su, X.-D, Taddei, N, Stefani, M, Ramponi, G, Nordlund, P.
登録日1994-07-05
公開日1995-07-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The crystal structure of a low-molecular-weight phosphotyrosine protein phosphatase.
Nature, 370, 1994
1GXT
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Hydrogenase Maturation Protein HypF "acylphosphatase-like" N-terminal domain (HypF-ACP) in complex with Sulfate
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, HYDROGENASE MATURATION PROTEIN HYPF, ...
著者Rosano, C, Zuccotti, S, Stefani, M, Bucciantini, M, Ramponi, G, Bolognesi, M.
登録日2002-04-11
公開日2002-09-12
最終更新日2019-07-24
実験手法X-RAY DIFFRACTION (1.27 Å)
主引用文献Crystal Structure and Anion Binding in the Prokaryotic Hydrogenase Maturation Factor Hypf Acylphosphatase-Like Domain
J.Mol.Biol., 321, 2002
1GXU
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Hydrogenase Maturation Protein HypF "acylphosphatase-like" N-terminal domain (HypF-ACP) in complex with a substrate. Crystal grown in the presence of carbamoylphosphate
分子名称: DIHYDROGENPHOSPHATE ION, HYDROGENASE MATURATION PROTEIN HYPF
著者Rosano, C, Zuccotti, S, Stefani, M, Bucciantini, M, Ramponi, G, Bolognesi, M.
登録日2002-04-11
公開日2002-09-12
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.27 Å)
主引用文献Crystal Structure and Anion Binding in the Prokaryotic Hydrogenase Maturation Factor Hypf Acylphosphatase-Like Domain
J.Mol.Biol., 321, 2002
2MYG
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Solution structure of the dithiolic glutaredoxin 2-C-Grx1 from the pathogen Trypanosoma brucei brucei
分子名称: Dithiol glutaredoxin 1
著者Sturlese, M, Stefani, M, Manta, B, Mammi, S, Comini, M, Bellanda, M.
登録日2015-01-22
公開日2016-02-10
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Solution structure of the dithiolic glutaredoxin 2-C-Grx1 from the pathogen Trypanosoma brucei brucei
To be Published
2YIX
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Triazolopyridine Inhibitors of p38
分子名称: 1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea, MITOGEN-ACTIVATED PROTEIN KINASE 14
著者Millan, D.S, Anderson, M, Bunnage, M.E, Burrows, J.L, Butcher, K.J, Dodd, P.G, Evans, T.J, Fairman, D.A, Han, s, Hughes, S.J, Irving, S.L, Kilty, I.C, Lemaitre, A, Lewthawaite, R.A, Mahke, A, Marr, E, Mathias, J.P, Philip, J, Phillips, C, Smith, R.T, Stefaniak, M.H, Yeadon, M.
登録日2011-05-17
公開日2011-11-30
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Design and Synthesis of Inhaled P38 Inhibitors for the Treatment of Chronic Obstructive Pulmonary Disease.
J.Med.Chem., 54, 2011
2YIS
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triazolopyridine inhibitors of p38 kinase.
分子名称: 1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1H-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}urea, 2-fluoro-4-[4-(4-fluorophenyl)-1H-pyrazol-3-yl]pyridine, MITOGEN-ACTIVATED PROTEIN KINASE 14
著者Millan, D.S, Anderson, M, Bazin, R, Bunnage, M.E, Burrows, J.L, Butcher, K.J, Dodd, P.G, Evans, T.J, Fairman, D.A, Hughes, S.J, Irving, S.L, Kilty, I.C, Lemaitre, A, Lewthwaite, R.A, Mahnke, A, Mathais, J.P, Philip, J, Phillips, C, Smith, R.T, Stefaniack, M.H, Yeadon, M.
登録日2011-05-16
公開日2011-11-30
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Design and Synthesis of Inhaled P38 Inhibitors for the Treatment of Chronic Obstructive Pulmonary Disease.
J.Med.Chem., 54, 2011

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