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PDB: 1 件

2X81
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BU of 2x81 by Molmil
STRUCTURE OF AURORA A IN COMPLEX WITH MLN8054
分子名称: 4-{[9-CHLORO-7-(2,6-DIFLUOROPHENYL)-5H-PYRIMIDO[5,4-D][2]BENZAZEPIN-2-YL]AMINO}BENZOIC ACID, SERINE/THREONINE-PROTEIN KINASE 6
著者Savory, W, Mueller, I, Mason, C.S, Lamers, M, Williams, D.H, Eyers, P.A.
登録日2010-03-05
公開日2010-05-05
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.91 Å)
主引用文献Drug-Resistant Aurora a Mutants for Cellular Target Validation of the Small Molecule Kinase Inhibitors Mln8054 and Mln8237.
Acs Chem.Biol., 5, 2010

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件を2024-07-17に公開中

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