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PDB: 53 results

7DI7
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BU of 7di7 by Molmil
Falcilysin in complex with chloroquine
Descriptor: ACETATE ION, Falcilysin, N4-(7-CHLORO-QUINOLIN-4-YL)-N1,N1-DIETHYL-PENTANE-1,4-DIAMINE, ...
Authors:Lin, J.Q, El Sahili, A, Lescar, J.
Deposit date:2020-11-18
Release date:2021-12-01
Last modified:2024-05-29
Method:X-RAY DIFFRACTION (1.82 Å)
Cite:Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development.
Cell Chem Biol, 31, 2024
7DIA
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BU of 7dia by Molmil
Falcilysin in complex with mefloquine
Descriptor: (S)-[2,8-bis(trifluoromethyl)quinolin-4-yl]-[(2S)-piperidin-2-yl]methanol, 1,2-ETHANEDIOL, ACETATE ION, ...
Authors:Lin, J.Q, El Sahili, A, Lescar, J.
Deposit date:2020-11-18
Release date:2021-12-01
Last modified:2024-05-29
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development.
Cell Chem Biol, 31, 2024
7VPE
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BU of 7vpe by Molmil
Falcilysin in complex with A1
Descriptor: (4S,5S)-1-[[3-[[(4S,5S)-4,5-diphenyl-4,5-dihydroimidazol-1-yl]methyl]phenyl]methyl]-4,5-diphenyl-4,5-dihydroimidazole, ACETATE ION, CHLORIDE ION, ...
Authors:Lin, J.Q, El Sahili, A, Lescar, J.
Deposit date:2021-10-16
Release date:2022-10-19
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (1.62 Å)
Cite:Title is not available yet as we are preparing the manuscript. Will update again once the paper is out.
To Be Published
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221051

건을2024-06-12부터공개중

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