6BQU
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![BU of 6bqu by Molmil](/molmil-images/mine/6bqu) | Human GR (418-507) in complex with monomeric DNA binding site | 分子名称: | DNA (5'-D(P*AP*AP*GP*CP*TP*AP*GP*TP*AP*CP*AP*TP*TP*TP*GP*C)-3'), DNA (5'-D(P*TP*GP*CP*AP*AP*AP*TP*GP*TP*AP*CP*TP*AP*GP*CP*T)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A. | 登録日 | 2017-11-28 | 公開日 | 2018-12-05 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | General and sequence-specific roles for DNA in glucocorticoid receptor DNA-binding stoichiometry To Be Published
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6BSF
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![BU of 6bsf by Molmil](/molmil-images/mine/6bsf) | Human GR (418-507) in complex with monomeric DNA binding site | 分子名称: | DNA (5'-D(P*AP*AP*GP*CP*TP*AP*GP*TP*AP*CP*AP*TP*TP*TP*GP*C)-3'), DNA (5'-D(P*TP*GP*CP*AP*AP*AP*TP*GP*TP*AP*CP*TP*AP*GP*CP*T)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A. | 登録日 | 2017-12-02 | 公開日 | 2018-12-05 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | General and sequence-specific roles for DNA in glucocorticoid receptor DNA-binding stoichiometry To Be Published
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6BSE
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![BU of 6bse by Molmil](/molmil-images/mine/6bse) | Glucocorticoid receptor bound to high cooperativity monomer sequence | 分子名称: | DNA (5'-D(P*AP*CP*CP*AP*CP*GP*TP*GP*TP*AP*CP*TP*TP*TP*TP*T)-3'), DNA (5'-D(P*TP*AP*AP*AP*AP*AP*GP*TP*AP*CP*AP*CP*GP*TP*GP*G)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A. | 登録日 | 2017-12-02 | 公開日 | 2018-12-05 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | General and sequence-specific roles for DNA in glucocorticoid receptor DNA-binding stoichiometry To Be Published
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3G6T
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![BU of 3g6t by Molmil](/molmil-images/mine/3g6t) | GR gamma DNA-binding domain:FKBP5 16bp complex-34 | 分子名称: | DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*GP*GP*GP*TP*GP*TP*TP*CP*T)-3'), DNA (5'-D(*TP*AP*GP*AP*AP*CP*AP*CP*CP*CP*TP*GP*TP*TP*CP*T)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-08 | 公開日 | 2009-04-21 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G9M
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![BU of 3g9m by Molmil](/molmil-images/mine/3g9m) | GR DNA-binding domain:Sgk 16bp complex-44 | 分子名称: | 1,2-ETHANEDIOL, DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*TP*TP*GP*TP*CP*CP*G)-3'), DNA (5'-D(*TP*CP*GP*GP*AP*CP*AP*AP*AP*AP*TP*GP*TP*TP*CP*T)-3'), ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-13 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.61 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G6P
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![BU of 3g6p by Molmil](/molmil-images/mine/3g6p) | GR DNA binding domain:FKBP5 complex, 18bp | 分子名称: | ACETATE ION, DNA (5'-D(*CP*CP*AP*GP*AP*AP*CP*AP*CP*CP*CP*TP*GP*TP*TP*CP*TP*G)-3'), DNA (5'-D(*CP*CP*AP*GP*AP*AP*CP*AP*GP*GP*GP*TP*GP*TP*TP*CP*TP*G)-3'), ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-07 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.985 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G6R
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![BU of 3g6r by Molmil](/molmil-images/mine/3g6r) | GR DNA binding domain:FKBP5 complex-52, 18bp | 分子名称: | DNA (5'-D(*CP*CP*AP*GP*AP*AP*CP*AP*CP*CP*CP*TP*GP*TP*TP*CP*TP*G)-3'), DNA (5'-D(*CP*CP*AP*GP*AP*AP*CP*AP*GP*GP*GP*TP*GP*TP*TP*CP*TP*G)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-08 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G6Q
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![BU of 3g6q by Molmil](/molmil-images/mine/3g6q) | GR DNA binding domain:FKBP5 binding site complex-9 | 分子名称: | DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*CP*CP*CP*TP*GP*TP*TP*CP*T)-3'), DNA (5'-D(*TP*AP*GP*AP*AP*CP*AP*GP*GP*GP*TP*GP*TP*TP*CP*T)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-08 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.26 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G8X
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![BU of 3g8x by Molmil](/molmil-images/mine/3g8x) | GR DNA binding domain:GilZ 16bp complex-65 | 分子名称: | 1,2-ETHANEDIOL, DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*GP*GP*GP*TP*TP*CP*C)-3'), DNA (5'-D(*TP*GP*GP*AP*AP*CP*CP*CP*AP*AP*TP*GP*TP*TP*CP*T)-3'), ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-12 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G9J
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![BU of 3g9j by Molmil](/molmil-images/mine/3g9j) | GR DNA binding domain:Pal, 18bp complex-36 | 分子名称: | 1,2-ETHANEDIOL, DNA (5'-D(*CP*CP*AP*GP*AP*AP*CP*AP*AP*AP*AP*TP*GP*TP*TP*CP*TP*G)-3'), DNA (5'-D(*CP*CP*AP*GP*AP*AP*CP*AP*TP*TP*TP*TP*GP*TP*TP*CP*TP*G)-3'), ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-13 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.32 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3FYL
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![BU of 3fyl by Molmil](/molmil-images/mine/3fyl) | GR DNA binding domain:CGT complex | 分子名称: | 1,2-ETHANEDIOL, DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*TP*TP*GP*TP*CP*CP*G)-3'), DNA (5'-D(*TP*CP*GP*GP*AP*CP*AP*AP*AP*AP*TP*GP*TP*TP*CP*T)-3'), ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-01-22 | 公開日 | 2009-04-21 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G9O
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![BU of 3g9o by Molmil](/molmil-images/mine/3g9o) | GR DNA-binding domain:Sgk 16bp complex-9 | 分子名称: | DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*TP*TP*GP*TP*CP*CP*G)-3'), DNA (5'-D(*TP*CP*GP*GP*AP*CP*AP*AP*AP*AP*TP*GP*TP*TP*CP*T)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-13 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G97
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![BU of 3g97 by Molmil](/molmil-images/mine/3g97) | GR DNA-binding domain:GilZ 16bp complex-9 | 分子名称: | 1,2-ETHANEDIOL, DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*GP*GP*GP*TP*TP*CP*C)-3'), DNA (5'-D(*TP*GP*GP*AP*AP*CP*CP*CP*AP*AP*TP*GP*TP*TP*CP*T)-3'), ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-13 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G99
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![BU of 3g99 by Molmil](/molmil-images/mine/3g99) | GR DNA binding domain:Pal complex-9 | 分子名称: | 1,2-ETHANEDIOL, BROMIDE ION, DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*TP*TP*GP*TP*TP*CP*T)-3'), ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-13 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G9P
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![BU of 3g9p by Molmil](/molmil-images/mine/3g9p) | GR DNA binding domain:Sgk 16bp complex-7 | 分子名称: | DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*TP*TP*GP*TP*CP*CP*G)-3'), DNA (5'-D(*TP*CP*GP*GP*AP*CP*AP*AP*AP*AP*TP*GP*TP*TP*CP*T)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-13 | 公開日 | 2009-04-14 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.652 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G9I
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![BU of 3g9i by Molmil](/molmil-images/mine/3g9i) | GR DNA Binding domain: Pal complex-35 | 分子名称: | 1,2-ETHANEDIOL, DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*TP*TP*GP*TP*TP*CP*T)-3'), DNA (5'-D(*TP*AP*GP*AP*AP*CP*AP*AP*AP*AP*TP*GP*TP*TP*CP*T)-3'), ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-13 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G6U
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![BU of 3g6u by Molmil](/molmil-images/mine/3g6u) | GR DNA-binding domain:FKBP5 16bp complex-49 | 分子名称: | DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*CP*CP*CP*TP*GP*TP*TP*CP*T)-3'), DNA (5'-D(*TP*AP*GP*AP*AP*CP*AP*GP*GP*GP*TP*GP*TP*TP*CP*T)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-08 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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3G8U
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![BU of 3g8u by Molmil](/molmil-images/mine/3g8u) | DNA binding domain:GilZ 16bp complex-5 | 分子名称: | DNA (5'-D(*AP*AP*GP*AP*AP*CP*AP*TP*TP*GP*GP*GP*TP*TP*CP*C)-3'), DNA (5'-D(*TP*GP*GP*AP*AP*CP*CP*CP*AP*AP*TP*GP*TP*TP*CP*T)-3'), Glucocorticoid receptor, ... | 著者 | Pufall, M.A, Yamamoto, K.R, Meijsing, S.H. | 登録日 | 2009-02-12 | 公開日 | 2009-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | DNA binding site sequence directs glucocorticoid receptor structure and activity. Science, 324, 2009
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1R36
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![BU of 1r36 by Molmil](/molmil-images/mine/1r36) | NMR-based structure of autoinhibited murine Ets-1 deltaN301 | 分子名称: | C-ets-1 protein | 著者 | Lee, G.M, Donaldson, L.W, Pufall, M.A, Kang, H.-S, Pot, I, Graves, B.J, McIntosh, L.P. | 登録日 | 2003-09-30 | 公開日 | 2004-11-09 | 最終更新日 | 2024-05-08 | 実験手法 | SOLUTION NMR | 主引用文献 | The Structural and Dynamic Basis of Ets-1 DNA Binding Autoinhibition J.Biol.Chem., 280, 2005
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1MDM
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![BU of 1mdm by Molmil](/molmil-images/mine/1mdm) | INHIBITED FRAGMENT OF ETS-1 AND PAIRED DOMAIN OF PAX5 BOUND TO DNA | 分子名称: | C-ETS-1 PROTEIN, PAIRED BOX PROTEIN PAX-5, PAX5/ETS BINDING SITE ON THE MB-1 PROMOTER | 著者 | Garvie, C.W, Pufall, M.A, Graves, B.J, Wolberger, C. | 登録日 | 2002-08-07 | 公開日 | 2002-12-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | STRUCTURAL ANALYSIS OF THE AUTOINHIBITION OF ETS-1 AND ITS ROLE IN PROTEIN PARTNERSHIPS J.Biol.Chem., 277, 2002
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1MD0
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![BU of 1md0 by Molmil](/molmil-images/mine/1md0) | |
4D9T
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![BU of 4d9t by Molmil](/molmil-images/mine/4d9t) | Rsk2 C-terminal Kinase Domain with inhibitor (E)-methyl 3-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl)-2-cyanoacrylate | 分子名称: | Ribosomal protein S6 kinase alpha-3, SODIUM ION, methyl (2S)-3-{4-amino-7-[(1E)-3-hydroxyprop-1-en-1-yl]-5-(4-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl}-2-cyanopropanoate | 著者 | Serafimova, I.M, Pufall, M.A, Krishnan, S, Duda, K, Cohen, M.S, Maglathlin, R.L, McFarland, J.M, Miller, R.M, Frodin, M, Taunton, J. | 登録日 | 2012-01-12 | 公開日 | 2012-04-25 | 最終更新日 | 2012-05-16 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Reversible targeting of noncatalytic cysteines with chemically tuned electrophiles. Nat.Chem.Biol., 8, 2012
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4D9U
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![BU of 4d9u by Molmil](/molmil-images/mine/4d9u) | Rsk2 C-terminal Kinase Domain, (E)-tert-butyl 3-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl)-2-cyanoacrylate | 分子名称: | Ribosomal protein S6 kinase alpha-3, SODIUM ION, tert-butyl (2S)-3-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyanopropanoate | 著者 | Serafimova, I.M, Pufall, M.A, Krishnan, S, Duda, K, Cohen, M.S, Maglathlin, R.L, McFarland, J.M, Miller, R.M, Frodin, M, Taunton, J. | 登録日 | 2012-01-12 | 公開日 | 2012-04-11 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Reversible targeting of noncatalytic cysteines with chemically tuned electrophiles. Nat.Chem.Biol., 8, 2012
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