3A0I
 
 | | Human glucokinase in complex with a synthetic activator | | 分子名称: | 3-[(4-fluorophenyl)sulfanyl]-N-(4-methyl-1,3-thiazol-2-yl)-6-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]pyridine-2-carboxamide, Glucokinase, SODIUM ION, ... | | 著者 | Kamata, K, Mitsuya, M. | | 登録日 | 2009-03-19 | | 公開日 | 2009-04-28 | | 最終更新日 | 2023-11-01 | | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | | 主引用文献 | Discovery of novel 3,6-disubstituted 2-pyridinecarboxamide derivatives as GK activators
Bioorg.Med.Chem.Lett., 19, 2009
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3GOI
 | | Human glucokinase in complex with a synthetic activator | | 分子名称: | 2-(methylamino)-N-(4-methyl-1,3-thiazol-2-yl)-5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]benzamide, Glucokinase, alpha-D-glucopyranose | | 著者 | Kamata, K, Mitsuya, M. | | 登録日 | 2009-03-19 | | 公開日 | 2009-04-28 | | 最終更新日 | 2024-03-20 | | 実験手法 | X-RAY DIFFRACTION (2.52 Å) | | 主引用文献 | Discovery of novel 3,6-disubstituted 2-pyridinecarboxamide derivatives as GK activators
Bioorg.Med.Chem.Lett., 19, 2009
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1V4T
 | | Crystal structure of human glucokinase | | 分子名称: | SODIUM ION, SULFATE ION, glucokinase isoform 2 | | 著者 | Kamata, K, Mitsuya, M, Nishimura, T, Eiki, J, Nagata, Y. | | 登録日 | 2003-11-19 | | 公開日 | 2004-03-30 | | 最終更新日 | 2023-11-08 | | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | | 主引用文献 | Structural basis for allosteric regulation of the monomeric allosteric enzyme human glucokinase
Structure, 12, 2004
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1V4S
 | | Crystal structure of human glucokinase | | 分子名称: | 2-AMINO-4-FLUORO-5-[(1-METHYL-1H-IMIDAZOL-2-YL)SULFANYL]-N-(1,3-THIAZOL-2-YL)BENZAMIDE, SODIUM ION, alpha-D-glucopyranose, ... | | 著者 | Kamata, K, Mitsuya, M, Nishimura, T, Eiki, J, Nagata, Y. | | 登録日 | 2003-11-19 | | 公開日 | 2004-03-30 | | 最終更新日 | 2023-11-08 | | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | | 主引用文献 | Structural basis for allosteric regulation of the monomeric allosteric enzyme human glucokinase
Structure, 12, 2004
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