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PDB: 83 件

3I2Z
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BU of 3i2z by Molmil
Structure of cold shock protein E from Salmonella typhimurium
分子名称: RNA chaperone, negative regulator of cspA transcription
著者Morgan, H.P, McNae, I, Wear, M.A, Gallagher, M, Walkinshaw, M.D.
登録日2009-06-30
公開日2009-12-22
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Crystallization and X-ray structure of cold-shock protein E from Salmonella typhimurium
Acta Crystallogr.,Sect.F, 65, 2009
3QV9
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BU of 3qv9 by Molmil
Crystal structure of Trypanosoma cruzi pyruvate kinase(TcPYK)in complex with ponceau S.
分子名称: 3-hydroxy-4-[(E)-{2-sulfo-4-[(E)-(4-sulfophenyl)diazenyl]phenyl}diazenyl]naphthalene-2,7-disulfonic acid, PHOSPHATE ION, POTASSIUM ION, ...
著者Morgan, H.P, Auld, D.S, McNae, I.W, Nowicki, M.W, Michels, P.A.M, Fothergill-Gilmore, L.A, Walkinshaw, M.D.
登録日2011-02-25
公開日2011-07-06
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The trypanocidal drug suramin and other trypan blue mimetics are inhibitors of pyruvate kinases and bind to the adenosine site.
J.Biol.Chem., 286, 2011
3SRK
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BU of 3srk by Molmil
A new class of suicide inhibitor blocks nucleotide binding to pyruvate kinase
分子名称: 1,2-BENZISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDE, POTASSIUM ION, Pyruvate kinase, ...
著者Morgan, H.P, Walsh, M, Blackburn, E.A, Wear, M.A, Boxer, M, Shen, M, McNae, I.W, Michels, P.A.M, Auld, D.S, Fothergill-Gilmore, L.A, Walkinshaw, M.D.
登録日2011-07-07
公開日2012-07-18
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献A new class of suicide inhibitor blocks nucleotide binding to pyruvate kinase
To be Published
4KRZ
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BU of 4krz by Molmil
Apo crystal structure of pyruvate kinase (PYK) from Trypanosoma cruzi
分子名称: GLYCEROL, POTASSIUM ION, Pyruvate kinase
著者Zhong, W, Morgan, H.P, McNae, I.W, Michels, P.A.M, Fothergill-Gilmore, L.A, Walkinshaw, M.D.
登録日2013-05-17
公開日2014-11-19
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structures of pyruvate kinases display evolutionarily divergent allosteric strategies.
R Soc Open Sci, 1, 2014
3SRF
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BU of 3srf by Molmil
Human M1 pyruvate kinase
分子名称: GLYCEROL, MAGNESIUM ION, PHOSPHATE ION, ...
著者Morgan, H.P, O'Reilly, F, Palmer, R, McNae, I.W, Nowicki, M.W, Wear, M.A, Fothergill-Gilmore, L.A, Walkinshaw, M.D.
登録日2011-07-07
公開日2012-08-08
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.845 Å)
主引用文献Allosetric regulation of M2 pyruvate kinase.
To be Published
3SRH
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BU of 3srh by Molmil
Human M2 pyruvate kinase
分子名称: PHOSPHATE ION, Pyruvate kinase isozymes M1/M2
著者Morgan, H.P, O'Reilly, F, Palmer, R, McNae, I.W, Nowicki, M.W, Wear, M.A, Fothergill-Gilmore, L.A, Walkinshaw, M.D.
登録日2011-07-07
公開日2012-08-08
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Allosetric regulation of M2 pyruvate kinase.
To be Published
3SRD
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BU of 3srd by Molmil
Human M2 pyruvate kinase in complex with fructose 1-6 bisphosphate and Oxalate.
分子名称: 1,6-di-O-phosphono-beta-D-fructofuranose, GLYCEROL, MAGNESIUM ION, ...
著者Morgan, H.P, O'Reilly, F, Palmer, R, McNae, I.W, Nowicki, M.W, Wear, M.A, Fothergill-Gilmore, L.A, Walkinshaw, M.D.
登録日2011-07-07
公開日2012-08-08
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.902 Å)
主引用文献Allosetric regulation of M2 pyruvate kinase.
To be Published
5OEZ
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BU of 5oez by Molmil
Crystal structure of Leishmania major fructose-1,6-bisphosphatase in apo form.
分子名称: FBP protein
著者Yuan, M, Vasquez-Valdivieso, M.G, McNae, I.W, Michels, P.A.M, Fothergill-Gilmore, L.A, Walkinshaw, M.D.
登録日2017-07-10
公開日2017-09-20
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献Structures of Leishmania Fructose-1,6-Bisphosphatase Reveal Species-Specific Differences in the Mechanism of Allosteric Inhibition.
J. Mol. Biol., 429, 2017
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