Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 264 results

5M7E
DownloadVisualize
BU of 5m7e by Molmil
Tubulin-BKM120 complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amine, CALCIUM ION, ...
Authors:Bohnacker, T, Prota, A.E, Steinmetz, M.O, Wymann, M.P.
Deposit date:2016-10-27
Release date:2017-02-22
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.046 Å)
Cite:Deconvolution of Buparlisib's mechanism of action defines specific PI3K and tubulin inhibitors for therapeutic intervention.
Nat Commun, 8, 2017
5NQU
DownloadVisualize
BU of 5nqu by Molmil
Tubulin Darpin cryo structure
Descriptor: Designed Ankyrin Repeat Protein (DARPIN) D1, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
Authors:Weinert, T, Olieric, N, James, D, Gashi, D, Nogly, P, Jaeger, K, Steinmetz, M.O, Standfuss, J.
Deposit date:2017-04-21
Release date:2017-09-27
Last modified:2024-05-08
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Serial millisecond crystallography for routine room-temperature structure determination at synchrotrons.
Nat Commun, 8, 2017
5M5C
DownloadVisualize
BU of 5m5c by Molmil
Mechanism of microtubule minus-end recognition and protection by CAMSAP proteins
Descriptor: Calmodulin-regulated spectrin-associated protein 1, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
Authors:Akhmanova, A, Moores, C.A, Baldus, M, Steinmetz, M.O, Topf, M, Roberts, A.J, Grant, B.J, Scarabelli, G, Joseph, A.-P, van Hooff, J.J.E, Houben, K, Hua, S, Luo, Y, Stangier, M.M, Jiang, K, Atherton, J.
Deposit date:2016-10-21
Release date:2017-10-04
Last modified:2024-05-15
Method:ELECTRON MICROSCOPY (4.8 Å)
Cite:A structural model for microtubule minus-end recognition and protection by CAMSAP proteins.
Nat. Struct. Mol. Biol., 24, 2017
5M50
DownloadVisualize
BU of 5m50 by Molmil
Mechanism of microtubule minus-end recognition and protection by CAMSAP proteins
Descriptor: Calmodulin-regulated spectrin-associated protein 3, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
Authors:Akhmanova, A, Moores, C.A, Baldus, M, Steinmetz, M.O, Topf, M, Roberts, A.J, Grant, B.J, Scarabelli, G, Joseph, A.-P, van Hooff, J.J.E, Houben, K, Hua, S, Luo, Y, Stangier, M.M, Jiang, K, Atherton, J.
Deposit date:2016-10-20
Release date:2017-10-04
Last modified:2024-05-15
Method:ELECTRON MICROSCOPY (5.3 Å)
Cite:A structural model for microtubule minus-end recognition and protection by CAMSAP proteins.
Nat. Struct. Mol. Biol., 24, 2017
5M7G
DownloadVisualize
BU of 5m7g by Molmil
Tubulin-MTD147 complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5-(2,6-dimorpholin-4-ylpyridin-4-yl)-4-(trifluoromethyl)pyridin-2-amine, CALCIUM ION, ...
Authors:Bohnacker, T, Prota, A.E, Steinmetz, M.O, Wymann, M.P.
Deposit date:2016-10-27
Release date:2017-02-22
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.248 Å)
Cite:Deconvolution of Buparlisib's mechanism of action defines specific PI3K and tubulin inhibitors for therapeutic intervention.
Nat Commun, 8, 2017
5M8D
DownloadVisualize
BU of 5m8d by Molmil
Tubulin MTD265-R1 complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5-(6-morpholin-4-yl-2-pyrrolidin-1-yl-pyrimidin-4-yl)-4-(trifluoromethyl)pyridin-2-amine, CALCIUM ION, ...
Authors:Bohnacker, T, Prota, A.E, Steinmetz, M.O, Wymann, M.P.
Deposit date:2016-10-28
Release date:2017-03-22
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:Deconvolution of Buparlisib's mechanism of action defines specific PI3K and tubulin inhibitors for therapeutic intervention.
Nat Commun, 8, 2017
6RJ8
DownloadVisualize
BU of 6rj8 by Molmil
Structure of the alpha-beta hydrolase CorS from Tabernathe iboga
Descriptor: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, TETRAETHYLENE GLYCOL, ...
Authors:Farrow, S.C, Caputi, L, Kamileen, M.O, Bussey, K, Stevenson, C.E.M, Mundy, J, Lawson, D.M, O'Connor, S.E.
Deposit date:2019-04-26
Release date:2020-03-04
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.42 Å)
Cite:Structural basis of cycloaddition in biosynthesis of iboga and aspidosperma alkaloids.
Nat.Chem.Biol., 16, 2020
5S53
DownloadVisualize
BU of 5s53 by Molmil
Tubulin-Z1349163663-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 6-[cyclobutyl(methyl)amino]pyridazine-3-carboxamide, CALCIUM ION, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.75 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5Q
DownloadVisualize
BU of 5s5q by Molmil
Tubulin-Z396380540-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.05 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S54
DownloadVisualize
BU of 5s54 by Molmil
Tubulin-Z2856434816-complex
Descriptor: 1-(pyridin-4-yl)-N-[(thiophen-2-yl)methyl]methanamine, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5T
DownloadVisualize
BU of 5s5t by Molmil
Tubulin-Z198194394-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-(4-fluorophenyl)piperazine-1-carboxamide, CALCIUM ION, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.53 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S55
DownloadVisualize
BU of 5s55 by Molmil
Tubulin-Z106307058-complex
Descriptor: 2-methyl-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S67
DownloadVisualize
BU of 5s67 by Molmil
Tubulin-Z1896597864-complex
Descriptor: 1-(6-methoxypyridin-2-yl)-N-methylmethanamine, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S56
DownloadVisualize
BU of 5s56 by Molmil
Tubulin-Z2856434783-complex
Descriptor: CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5V
DownloadVisualize
BU of 5s5v by Molmil
Tubulin-Z32386228-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5-chloranyl-2-methoxy-~{N}-(2-methylpropyl)benzamide, CALCIUM ION, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S58
DownloadVisualize
BU of 5s58 by Molmil
Tubulin-Z2856434826-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S57
DownloadVisualize
BU of 5s57 by Molmil
Tubulin-Z2856434883-complex
Descriptor: 1-{4-[(2-phenylethyl)amino]piperidin-1-yl}ethan-1-one, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.45 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5S
DownloadVisualize
BU of 5s5s by Molmil
Tubulin-Z166605480-complex
Descriptor: (1S)-1-(4-fluorophenyl)-N-methylethan-1-amine, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.36 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S59
DownloadVisualize
BU of 5s59 by Molmil
Tubulin-Z1324080698-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 3-fluoro-5-methylbenzene-1-sulfonamide, CALCIUM ION, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5W
DownloadVisualize
BU of 5s5w by Molmil
Tubulin-Z53860899-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5D
DownloadVisualize
BU of 5s5d by Molmil
Tubulin-Z32400357-complex
Descriptor: 1-(3-methylbenzene-1-carbonyl)piperidine-4-carboxamide, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5U
DownloadVisualize
BU of 5s5u by Molmil
Tubulin-Z1124201124-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5C
DownloadVisualize
BU of 5s5c by Molmil
Tubulin-Z44592329-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5X
DownloadVisualize
BU of 5s5x by Molmil
Tubulin-Z45705015-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.32 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021
5S5B
DownloadVisualize
BU of 5s5b by Molmil
Tubulin-Z906021418-complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5-chloro-2-(propan-2-yl)pyrimidine-4-carboxamide, CALCIUM ION, ...
Authors:Muehlethaler, T, Gioia, D, Prota, A.E, Sharpe, M.E, Cavalli, A, Steinmetz, M.O.
Deposit date:2020-11-08
Release date:2021-06-30
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Comprehensive Analysis of Binding Sites in Tubulin.
Angew.Chem.Int.Ed.Engl., 60, 2021

221051

數據於2024-06-12公開中

PDB statisticsPDBj update infoContact PDBjnumon