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PDB: 303 件

3QQ8
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Crystal structure of p97-N in complex with FAF1-UBX
分子名称: CHLORIDE ION, FAS-associated factor 1, Transitional endoplasmic reticulum ATPase
著者Haenzelmann, P, Schindelin, H.
登録日2011-02-15
公開日2011-06-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Hierarchical Binding of Cofactors to the AAA ATPase p97.
Structure, 19, 2011
4BX2
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BU of 4bx2 by Molmil
Crystal Structure of murine Chronophin (Pyridoxal Phosphate Phosphatase) in complex with Beryllium trifluoride
分子名称: BERYLLIUM TRIFLUORIDE ION, GLYCEROL, MAGNESIUM ION, ...
著者Knobloch, G, Gohla, A, Schindelin, H.
登録日2013-07-08
公開日2013-12-25
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.193 Å)
主引用文献Chronophin Dimerization is Required for Proper Positioning of its Substrate Specificity Loop.
J.Biol.Chem., 289, 2014
2RDI
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Snapshots of a Y-family DNA polymerase in replication: Dpo4 in apo and binary/ternary complex forms
分子名称: DI(HYDROXYETHYL)ETHER, DNA polymerase IV, GLYCEROL
著者Wong, J.H.Y, Ling, H.
登録日2007-09-24
公開日2008-06-24
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Snapshots of a Y-family DNA polymerase in replication: substrate-induced conformational transitions and implications for fidelity of Dpo4.
J.Mol.Biol., 379, 2008
3R3M
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Crystal structure of the FAF1 UBX domain
分子名称: FAS-associated factor 1, PHOSPHATE ION
著者Haenzelmann, P, Schindelin, H.
登録日2011-03-16
公開日2011-06-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Hierarchical Binding of Cofactors to the AAA ATPase p97.
Structure, 19, 2011
4EYH
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Human DNA polymerase iota incorporating dCTP opposite N-(deoxyguanosin-8-yl)-1-aminopyrene lesion
分子名称: 2'-DEOXYCYTIDINE-5'-TRIPHOSPHATE, DNA polymerase iota, DNA primer, ...
著者Kirouac, K, Ling, H.
登録日2012-05-01
公開日2013-01-09
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Replication of a carcinogenic nitropyrene DNA lesion by human Y-family DNA polymerase.
Nucleic Acids Res., 41, 2013
1QZT
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Phosphotransacetylase from Methanosarcina thermophila
分子名称: Phosphate acetyltransferase, SULFATE ION
著者Iyer, P.P, Lawrence, S.H, Luther, K.B, Rajashankar, K.R, Yennawar, H.P, Ferry, J.G, Schindelin, H.
登録日2003-09-17
公開日2004-06-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of phosphotransacetylase from the methanogenic archaeon Methanosarcina thermophila.
STRUCTURE, 12, 2004
1FR9
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STRUCTURE OF E. COLI MOBA
分子名称: ACETATE ION, MOLYBDOPTERIN-GUANINE DINUCLEOTIDE BIOSYNTHESIS PROTEIN, ZINC ION
著者Lake, M.W, Temple, C.A, Rajagopalan, K.V, Schindelin, H.
登録日2000-09-07
公開日2001-01-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献The crystal structure of the Escherichia coli MobA protein provides insight into molybdopterin guanine dinucleotide biosynthesis.
J.Biol.Chem., 275, 2000
1FRW
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STRUCTURE OF E. COLI MOBA WITH BOUND GTP AND MANGANESE
分子名称: ACETATE ION, GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, ...
著者Lake, M.W, Temple, C.A, Rajagopalan, K.V, Schindelin, H.
登録日2000-09-07
公開日2001-01-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献The crystal structure of the Escherichia coli MobA protein provides insight into molybdopterin guanine dinucleotide biosynthesis.
J.Biol.Chem., 275, 2000
4GLJ
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Crystal structure of methylthioadenosine phosphorylase in complex with rhodamine B
分子名称: CHLORIDE ION, N-[9-(2-carboxyphenyl)-6-(diethylamino)-3H-xanthen-3-ylidene]-N-ethylethanaminium, PHOSPHATE ION, ...
著者Bujacz, A, Bujacz, G, Cieslinski, H, Bartasun, P.
登録日2012-08-14
公開日2013-02-20
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A study on the interaction of rhodamine B with methylthioadenosine phosphorylase protein sourced from an antarctic soil metagenomic library.
Plos One, 8, 2013
4F9Z
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Crystal Structure of human ERp27
分子名称: 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, 3,6,9,12,15,18,21,24,27,30,33,36,39-TRIDECAOXAHENTETRACONTANE-1,41-DIOL, ACETATE ION, ...
著者Kober, F.X, Koelmel, W, Kuper, J, Schindelin, H.
登録日2012-05-21
公開日2012-12-05
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Crystal Structure of the Protein-Disulfide Isomerase Family Member ERp27 Provides Insights into Its Substrate Binding Capabilities.
J.Biol.Chem., 288, 2013
1NVI
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Orthorhombic Crystal Form of Molybdopterin Synthase
分子名称: GLYCEROL, Molybdopterin converting factor subunit 1, Molybdopterin converting factor subunit 2, ...
著者Rudolph, M.J, Wuebbens, M.M, Turque, O, Rajagopalan, K.V, Schindelin, H.
登録日2003-02-03
公開日2003-05-06
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Studies of Molybdopterin Synthase Provide Insights into its Catalytic Mechanism
J.Biol.Chem., 278, 2003
4PD1
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BU of 4pd1 by Molmil
Structure of gephyrin E domain with Glycine-beta receptor peptide
分子名称: ACETATE ION, GLYCEROL, Gephyrin, ...
著者Kasaragod, V.B, Maric, H.M, Schindelin, H.
登録日2014-04-17
公開日2014-08-27
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.975 Å)
主引用文献Modulation of gephyrin-glycine receptor affinity by multivalency.
Acs Chem.Biol., 9, 2014
2FTS
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BU of 2fts by Molmil
Crystal structure of the glycine receptor-gephyrin complex
分子名称: Glycine receptor beta chain precursor, gephyrin
著者Kim, E.Y, Schindelin, H.
登録日2006-01-24
公開日2006-03-14
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献Deciphering the structural framework of glycine receptor anchoring by gephyrin.
Embo J., 25, 2006
4PD0
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BU of 4pd0 by Molmil
1.7 A resolution structure of gephyrin's E-domain
分子名称: Gephyrin
著者Kasaragod, V.B, Maric, H.M, Schindelin, H.
登録日2014-04-17
公開日2014-08-27
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Modulation of gephyrin-glycine receptor affinity by multivalency.
Acs Chem.Biol., 9, 2014
4FBU
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BU of 4fbu by Molmil
Dpo4 polymerase pre-insertion binary complex with the N-(deoxyguanosin-8-yl)-1-aminopyrene lesion
分子名称: CALCIUM ION, DNA polymerase IV, DNA primer, ...
著者Kirouac, K, Basu, A, Ling, H.
登録日2012-05-23
公開日2013-06-12
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural mechanism of replication stalling on a bulky amino-polycyclic aromatic hydrocarbon DNA adduct by a y family DNA polymerase.
J.Mol.Biol., 425, 2013
5T14
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DNA polymerase kappa extending beyond a bulky major benzo[a]pyrene adduct
分子名称: 2'-deoxy-5'-O-[(R)-hydroxy{[(R)-hydroxy(phosphonooxy)phosphoryl]amino}phosphoryl]adenosine, DNA, DNA polymerase kappa, ...
著者Jha, V.K, Ling, H.
登録日2016-08-17
公開日2016-12-21
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural basis of accurate replication beyond a bulky major benzo[a]pyrene adduct by human DNA polymerase kappa.
DNA Repair (Amst.), 49, 2017
5T27
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mPI3Kd IN COMPLEX WITH 5d
分子名称: 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{S})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
4NNJ
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Crystal structure of Uba1 in complex with ubiquitin-AMP and thioesterified ubiquitin
分子名称: ADENOSINE MONOPHOSPHATE, GLYCEROL, SULFATE ION, ...
著者Schaefer, A, Schindelin, H.
登録日2013-11-18
公開日2014-05-07
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of the ubiquitin-activating enzyme loaded with two ubiquitin molecules.
Acta Crystallogr.,Sect.D, 70, 2014
5T23
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PI3Kg IN COMPLEX WITH 5d
分子名称: 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{S})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.78 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
5T2B
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mPI3Kd IN COMPLEX WITH 5e
分子名称: 5-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]-3-(1~{H}-pyrazol-4-yl)pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
5T2I
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mPI3Kd IN COMPLEX WITH 7k
分子名称: 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-4-carboxamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
4FBT
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Dpo4 post-insertion complex with the N-(deoxyguanosin-8-yl)-1-aminopyrene lesion
分子名称: 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, CALCIUM ION, DNA polymerase IV, ...
著者Kirouac, K, Ling, H.
登録日2012-05-23
公開日2013-06-12
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural mechanism of replication stalling on a bulky amino-polycyclic aromatic hydrocarbon DNA adduct by a y family DNA polymerase.
J.Mol.Biol., 425, 2013
5T2D
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mPI3Kd IN COMPLEX WITH 7j
分子名称: 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]-~{N},~{N}-dimethyl-pyrazole-1-sulfonamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
5T2M
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mPI3Kd IN COMPLEX WITH 7m
分子名称: 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]benzamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
2G9G
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Crystal structure of His-tagged mouse PNGase C-terminal domain
分子名称: GLYCEROL, SULFATE ION, peptide N-glycanase
著者Zhou, X, Zhao, G, Wang, L, Li, G, Lennarz, W.J, Schindelin, H.
登録日2006-03-06
公開日2006-10-24
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and biochemical studies of the C-terminal domain of mouse peptide-N-glycanase identify it as a mannose-binding module.
Proc.Natl.Acad.Sci.Usa, 103, 2006

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