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Crystal Structure of PAK4 in complex with inhibitor 47
Descriptor:	Serine/threonine-protein kinase PAK 4, [(3R)-3-azanylpiperidin-1-yl]-[1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]methanone
Authors:	Zhao, F, Li, H.
Deposit date:	2020-08-05
Release date:	2021-08-11
Last modified:	2023-11-29
Method:	X-RAY DIFFRACTION (2.9 Å)
Cite:	Discovery of 6-ethynyl-1H-indole-3-carboxamide Derivatives as Highly Potent and Selective p21-Activated Kinase 4 (PAK4) Inhibitors to be published

Crystal Structure of PAK4 in complex with inhibitor 55
Descriptor:	Serine/threonine-protein kinase PAK 4, [1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]-[(3S)-3-methylpiperazin-1-yl]methanone
Authors:	Zhao, F, Li, H.
Deposit date:	2020-08-06
Release date:	2021-08-11
Last modified:	2023-11-29
Method:	X-RAY DIFFRACTION (2.5 Å)
Cite:	Discovery of 6-ethynyl-1H-indole-3-carboxamide Derivatives as Highly Potent and Selective p21-Activated Kinase 4 (PAK4) Inhibitors to be published