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PDB: 1777 件

7CP3
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BU of 7cp3 by Molmil
Crystal Structure of PAK4 in complex with inhibitor 47
分子名称: Serine/threonine-protein kinase PAK 4, [(3R)-3-azanylpiperidin-1-yl]-[1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]methanone
著者Zhao, F, Li, H.
登録日2020-08-05
公開日2021-08-11
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Discovery of 6-ethynyl-1H-indole-3-carboxamide Derivatives as Highly Potent and Selective p21-Activated Kinase 4 (PAK4) Inhibitors
to be published
7CP4
DownloadVisualize
BU of 7cp4 by Molmil
Crystal Structure of PAK4 in complex with inhibitor 55
分子名称: Serine/threonine-protein kinase PAK 4, [1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]-[(3S)-3-methylpiperazin-1-yl]methanone
著者Zhao, F, Li, H.
登録日2020-08-06
公開日2021-08-11
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Discovery of 6-ethynyl-1H-indole-3-carboxamide Derivatives as Highly Potent and Selective p21-Activated Kinase 4 (PAK4) Inhibitors
to be published

222036

件を2024-07-03に公開中

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