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PDB: 13 件

4IL3
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Crystal Structure of S. mikatae Ste24p
分子名称: Ste24p, ZINC ION
著者Pryor Jr, E.E, Horanyi, P.S, Clark, K, Fedoriw, N, Connelly, S.M, Koszelak-Rosenblum, M, Zhu, G, Malkowski, M.G, Dumont, M.E, Wiener, M.C, Membrane Protein Structural Biology Consortium (MPSBC)
登録日2012-12-28
公開日2013-02-20
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.102 Å)
主引用文献Structure of the integral membrane protein CAAX protease Ste24p.
Science, 339, 2013
7MF0
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Co-crystal structure of PERK with inhibitor (R)-2-amino-N-cyclopropyl-5-(4-(2-(3,5-difluorophenyl)-2-hydroxyacetamido)-2-methylphenyl)nicotinamide
分子名称: 2-amino-N-cyclopropyl-5-(4-{[(2R)-2-(3,5-difluorophenyl)-2-hydroxyacetyl]amino}-2-methylphenyl)pyridine-3-carboxamide, Eukaryotic translation initiation factor 2-alpha kinase 3,Eukaryotic translation initiation factor 2-alpha kinase 3
著者Wiens, B, Koszelak-Rosenblum, M, Surman, M.D, Zhu, G, Mulvihill, M.J.
登録日2021-04-08
公開日2021-05-19
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.809 Å)
主引用文献Discovery of 2-amino-3-amido-5-aryl-pyridines as highly potent, orally bioavailable, and efficacious PERK kinase inhibitors.
Bioorg.Med.Chem.Lett., 43, 2021
4ZR1
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Hydroxylase domain of scs7p
分子名称: Ceramide very long chain fatty acid hydroxylase SCS7, TRIDECANE, ZINC ION, ...
著者Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G, Membrane Protein Structural Biology Consortium (MPSBC)
登録日2015-05-11
公開日2015-07-29
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.6008 Å)
主引用文献The Crystal Structure of an Integral Membrane Fatty Acid alpha-Hydroxylase.
J.Biol.Chem., 290, 2015
4ZR0
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Full length scs7p (only hydroxylase domain visible)
分子名称: Ceramide very long chain fatty acid hydroxylase SCS7, ZINC ION
著者Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G, Membrane Protein Structural Biology Consortium (MPSBC)
登録日2015-05-11
公開日2015-07-29
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献The Crystal Structure of an Integral Membrane Fatty Acid alpha-Hydroxylase.
J.Biol.Chem., 290, 2015
4HHR
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Crystal Structure of fatty acid alpha-dioxygenase (Arabidopsis thaliana)
分子名称: Alpha-dioxygenase, CALCIUM ION, CHLORIDE ION, ...
著者Goulah, C.C, Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G.
登録日2012-10-10
公開日2013-02-20
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献The crystal structure of alpha-Dioxygenase provides insight into diversity in the cyclooxygenase-peroxidase superfamily.
Biochemistry, 52, 2013
4HHS
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Crystal Structure of fatty acid alpha-dioxygenase (Arabidopsis thaliana)
分子名称: Alpha-dioxygenase, CALCIUM ION, CHLORIDE ION, ...
著者Goulah, C.C, Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G.
登録日2012-10-10
公開日2013-02-20
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The crystal structure of alpha-Dioxygenase provides insight into diversity in the cyclooxygenase-peroxidase superfamily.
Biochemistry, 52, 2013
4KVJ
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Crystal structure of Oryza sativa fatty acid alpha-dioxygenase with hydrogen peroxide
分子名称: 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, CALCIUM ION, CHLORIDE ION, ...
著者Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G.
登録日2013-05-22
公開日2013-08-21
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Crystal structures of alpha-dioxygenase from Oryza sativa: Insights into substrate binding and activation by hydrogen peroxide.
Protein Sci., 22, 2013
4KVL
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Crystal structure of Oryza sativa fatty acid alpha-dioxygenase Y379F with palmitic acid
分子名称: CALCIUM ION, CHLORIDE ION, Fatty acid alpha-oxidase, ...
著者Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G.
登録日2013-05-22
公開日2013-08-21
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Crystal structures of alpha-dioxygenase from Oryza sativa: Insights into substrate binding and activation by hydrogen peroxide.
Protein Sci., 22, 2013
4KVK
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Crystal structure of Oryza sativa fatty acid alpha-dioxygenase
分子名称: CALCIUM ION, CHLORIDE ION, DECYL-BETA-D-MALTOPYRANOSIDE, ...
著者Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G.
登録日2013-05-22
公開日2013-08-21
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献Crystal structures of alpha-dioxygenase from Oryza sativa: Insights into substrate binding and activation by hydrogen peroxide.
Protein Sci., 22, 2013
3K8I
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Structure of crystal form IV of TP0453
分子名称: 30kLP
著者Zhu, G, Luthra, A, Desrosiers, D, Koszelak-Rosenblum, M, Mulay, V, Radolf, J.D, Malkowski, M.G.
登録日2009-10-14
公開日2010-10-27
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Transition from Closed to Open Conformation of Treponema pallidum Outer Membrane-associated Lipoprotein TP0453 Involves Membrane Sensing and Integration by Two Amphipathic Helices.
J.Biol.Chem., 286, 2011
3K8G
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Structure of crystal form I of TP0453
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 30kLP
著者Zhu, G, Luthra, A, Desrosiers, D, Koszelak-Rosenblum, M, Mulay, V, Radolf, J.D, Malkowski, M.G.
登録日2009-10-14
公開日2010-10-27
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献The Transition from Closed to Open Conformation of Treponema pallidum Outer Membrane-associated Lipoprotein TP0453 Involves Membrane Sensing and Integration by Two Amphipathic Helices.
J.Biol.Chem., 286, 2011
3K8H
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Structure of crystal form I of TP0453
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 30kLP
著者Zhu, G, Luthra, A, Desrosiers, D, Koszelak-Rosenblum, M, Mulay, V, Radolf, J.D, Malkowski, M.G.
登録日2009-10-14
公開日2010-10-27
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献The Transition from Closed to Open Conformation of Treponema pallidum Outer Membrane-associated Lipoprotein TP0453 Involves Membrane Sensing and Integration by Two Amphipathic Helices.
J.Biol.Chem., 286, 2011
3K8J
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Structure of crystal form III of TP0453
分子名称: 30kLP
著者Zhu, G, Luthra, A, Desrosiers, D, Koszelak-Rosenblum, M, Mulay, V, Radolf, J.D, Malkowski, M.G.
登録日2009-10-14
公開日2010-10-27
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Transition from Closed to Open Conformation of Treponema pallidum Outer Membrane-associated Lipoprotein TP0453 Involves Membrane Sensing and Integration by Two Amphipathic Helices.
J.Biol.Chem., 286, 2011

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