4IL3
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![BU of 4il3 by Molmil](/molmil-images/mine/4il3) | Crystal Structure of S. mikatae Ste24p | 分子名称: | Ste24p, ZINC ION | 著者 | Pryor Jr, E.E, Horanyi, P.S, Clark, K, Fedoriw, N, Connelly, S.M, Koszelak-Rosenblum, M, Zhu, G, Malkowski, M.G, Dumont, M.E, Wiener, M.C, Membrane Protein Structural Biology Consortium (MPSBC) | 登録日 | 2012-12-28 | 公開日 | 2013-02-20 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.102 Å) | 主引用文献 | Structure of the integral membrane protein CAAX protease Ste24p. Science, 339, 2013
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7MF0
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![BU of 7mf0 by Molmil](/molmil-images/mine/7mf0) | Co-crystal structure of PERK with inhibitor (R)-2-amino-N-cyclopropyl-5-(4-(2-(3,5-difluorophenyl)-2-hydroxyacetamido)-2-methylphenyl)nicotinamide | 分子名称: | 2-amino-N-cyclopropyl-5-(4-{[(2R)-2-(3,5-difluorophenyl)-2-hydroxyacetyl]amino}-2-methylphenyl)pyridine-3-carboxamide, Eukaryotic translation initiation factor 2-alpha kinase 3,Eukaryotic translation initiation factor 2-alpha kinase 3 | 著者 | Wiens, B, Koszelak-Rosenblum, M, Surman, M.D, Zhu, G, Mulvihill, M.J. | 登録日 | 2021-04-08 | 公開日 | 2021-05-19 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.809 Å) | 主引用文献 | Discovery of 2-amino-3-amido-5-aryl-pyridines as highly potent, orally bioavailable, and efficacious PERK kinase inhibitors. Bioorg.Med.Chem.Lett., 43, 2021
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4ZR1
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![BU of 4zr1 by Molmil](/molmil-images/mine/4zr1) | Hydroxylase domain of scs7p | 分子名称: | Ceramide very long chain fatty acid hydroxylase SCS7, TRIDECANE, ZINC ION, ... | 著者 | Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G, Membrane Protein Structural Biology Consortium (MPSBC) | 登録日 | 2015-05-11 | 公開日 | 2015-07-29 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.6008 Å) | 主引用文献 | The Crystal Structure of an Integral Membrane Fatty Acid alpha-Hydroxylase. J.Biol.Chem., 290, 2015
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4ZR0
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4HHR
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![BU of 4hhr by Molmil](/molmil-images/mine/4hhr) | Crystal Structure of fatty acid alpha-dioxygenase (Arabidopsis thaliana) | 分子名称: | Alpha-dioxygenase, CALCIUM ION, CHLORIDE ION, ... | 著者 | Goulah, C.C, Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G. | 登録日 | 2012-10-10 | 公開日 | 2013-02-20 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.51 Å) | 主引用文献 | The crystal structure of alpha-Dioxygenase provides insight into diversity in the cyclooxygenase-peroxidase superfamily. Biochemistry, 52, 2013
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4HHS
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![BU of 4hhs by Molmil](/molmil-images/mine/4hhs) | Crystal Structure of fatty acid alpha-dioxygenase (Arabidopsis thaliana) | 分子名称: | Alpha-dioxygenase, CALCIUM ION, CHLORIDE ION, ... | 著者 | Goulah, C.C, Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G. | 登録日 | 2012-10-10 | 公開日 | 2013-02-20 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The crystal structure of alpha-Dioxygenase provides insight into diversity in the cyclooxygenase-peroxidase superfamily. Biochemistry, 52, 2013
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4KVJ
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![BU of 4kvj by Molmil](/molmil-images/mine/4kvj) | Crystal structure of Oryza sativa fatty acid alpha-dioxygenase with hydrogen peroxide | 分子名称: | 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, CALCIUM ION, CHLORIDE ION, ... | 著者 | Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G. | 登録日 | 2013-05-22 | 公開日 | 2013-08-21 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.12 Å) | 主引用文献 | Crystal structures of alpha-dioxygenase from Oryza sativa: Insights into substrate binding and activation by hydrogen peroxide. Protein Sci., 22, 2013
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4KVL
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![BU of 4kvl by Molmil](/molmil-images/mine/4kvl) | Crystal structure of Oryza sativa fatty acid alpha-dioxygenase Y379F with palmitic acid | 分子名称: | CALCIUM ION, CHLORIDE ION, Fatty acid alpha-oxidase, ... | 著者 | Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G. | 登録日 | 2013-05-22 | 公開日 | 2013-08-21 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | Crystal structures of alpha-dioxygenase from Oryza sativa: Insights into substrate binding and activation by hydrogen peroxide. Protein Sci., 22, 2013
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4KVK
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![BU of 4kvk by Molmil](/molmil-images/mine/4kvk) | Crystal structure of Oryza sativa fatty acid alpha-dioxygenase | 分子名称: | CALCIUM ION, CHLORIDE ION, DECYL-BETA-D-MALTOPYRANOSIDE, ... | 著者 | Zhu, G, Koszelak-Rosenblum, M, Malkowski, M.G. | 登録日 | 2013-05-22 | 公開日 | 2013-08-21 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Crystal structures of alpha-dioxygenase from Oryza sativa: Insights into substrate binding and activation by hydrogen peroxide. Protein Sci., 22, 2013
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3K8I
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![BU of 3k8i by Molmil](/molmil-images/mine/3k8i) | Structure of crystal form IV of TP0453 | 分子名称: | 30kLP | 著者 | Zhu, G, Luthra, A, Desrosiers, D, Koszelak-Rosenblum, M, Mulay, V, Radolf, J.D, Malkowski, M.G. | 登録日 | 2009-10-14 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The Transition from Closed to Open Conformation of Treponema pallidum Outer Membrane-associated Lipoprotein TP0453 Involves Membrane Sensing and Integration by Two Amphipathic Helices. J.Biol.Chem., 286, 2011
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3K8G
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![BU of 3k8g by Molmil](/molmil-images/mine/3k8g) | Structure of crystal form I of TP0453 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 30kLP | 著者 | Zhu, G, Luthra, A, Desrosiers, D, Koszelak-Rosenblum, M, Mulay, V, Radolf, J.D, Malkowski, M.G. | 登録日 | 2009-10-14 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | The Transition from Closed to Open Conformation of Treponema pallidum Outer Membrane-associated Lipoprotein TP0453 Involves Membrane Sensing and Integration by Two Amphipathic Helices. J.Biol.Chem., 286, 2011
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3K8H
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![BU of 3k8h by Molmil](/molmil-images/mine/3k8h) | Structure of crystal form I of TP0453 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 30kLP | 著者 | Zhu, G, Luthra, A, Desrosiers, D, Koszelak-Rosenblum, M, Mulay, V, Radolf, J.D, Malkowski, M.G. | 登録日 | 2009-10-14 | 公開日 | 2010-10-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | The Transition from Closed to Open Conformation of Treponema pallidum Outer Membrane-associated Lipoprotein TP0453 Involves Membrane Sensing and Integration by Two Amphipathic Helices. J.Biol.Chem., 286, 2011
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3K8J
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![BU of 3k8j by Molmil](/molmil-images/mine/3k8j) | Structure of crystal form III of TP0453 | 分子名称: | 30kLP | 著者 | Zhu, G, Luthra, A, Desrosiers, D, Koszelak-Rosenblum, M, Mulay, V, Radolf, J.D, Malkowski, M.G. | 登録日 | 2009-10-14 | 公開日 | 2010-10-27 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The Transition from Closed to Open Conformation of Treponema pallidum Outer Membrane-associated Lipoprotein TP0453 Involves Membrane Sensing and Integration by Two Amphipathic Helices. J.Biol.Chem., 286, 2011
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