5RJY
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![BU of 5rjy by Molmil](/molmil-images/mine/5rjy) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z383325512 | Descriptor: | N-[(1H-pyrazol-4-yl)methyl]acetamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.25 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKE
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![BU of 5rke by Molmil](/molmil-images/mine/5rke) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z906021418 | Descriptor: | 5-chloro-2-(propan-2-yl)pyrimidine-4-carboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.291 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKS
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![BU of 5rks by Molmil](/molmil-images/mine/5rks) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1696844792 | Descriptor: | 1-(diphenylmethyl)azetidin-3-ol, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.24 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJK
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![BU of 5rjk by Molmil](/molmil-images/mine/5rjk) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024661 | Descriptor: | 5-bromo-2-hydroxybenzonitrile, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.21 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RK0
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![BU of 5rk0 by Molmil](/molmil-images/mine/5rk0) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z30932204 | Descriptor: | N-[(4-sulfamoylphenyl)methyl]acetamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.24 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKG
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![BU of 5rkg by Molmil](/molmil-images/mine/5rkg) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1124201124 | Descriptor: | PH-interacting protein, ethyl 1~{H}-pyrazole-4-carboxylate | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.282 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKW
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![BU of 5rkw by Molmil](/molmil-images/mine/5rkw) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z27678561 | Descriptor: | N-(6-methoxy-1,3-benzothiazol-2-yl)cyclopropanecarboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.242 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJZ
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![BU of 5rjz by Molmil](/molmil-images/mine/5rjz) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z755044716 | Descriptor: | N-ethyl-1H-1,2,3-triazole-4-carboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.275 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKF
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![BU of 5rkf by Molmil](/molmil-images/mine/5rkf) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1674937530 | Descriptor: | 2-(1-ethyl-1H-pyrazol-4-yl)ethan-1-ol, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.264 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKV
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![BU of 5rkv by Molmil](/molmil-images/mine/5rkv) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z56877838 | Descriptor: | 2-(4-ethoxyphenyl)ethanoic acid, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.277 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJU
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![BU of 5rju by Molmil](/molmil-images/mine/5rju) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z57261895 | Descriptor: | 2-cyclohexyl-N-(4H-1,2,4-triazol-4-yl)acetamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.32 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKA
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![BU of 5rka by Molmil](/molmil-images/mine/5rka) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z126932614 | Descriptor: | 2-[(methylsulfonyl)methyl]-1H-benzimidazole, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.33 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKO
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![BU of 5rko by Molmil](/molmil-images/mine/5rko) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z30620520 | Descriptor: | PH-interacting protein, cyclopropyl-[4-(4-fluorophenyl)piperazin-1-yl]methanone | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.42 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKY
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![BU of 5rky by Molmil](/molmil-images/mine/5rky) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1796014543 | Descriptor: | 1-[(2-fluorophenyl)methyl]-N-methylcyclopropane-1-carboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.38 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJT
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![BU of 5rjt by Molmil](/molmil-images/mine/5rjt) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z404993336 | Descriptor: | 5-methyl-N-(1-methyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.169 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RK8
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![BU of 5rk8 by Molmil](/molmil-images/mine/5rk8) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z53116498 | Descriptor: | 3-(2-methyl-1H-benzimidazol-1-yl)propanamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.272 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKJ
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![BU of 5rkj by Molmil](/molmil-images/mine/5rkj) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z373768898 | Descriptor: | N-(1-ethyl-1H-pyrazol-4-yl)cyclopentanecarboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.46 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJL
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![BU of 5rjl by Molmil](/molmil-images/mine/5rjl) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024662 | Descriptor: | (4-bromo-2-methoxyphenyl)methanol, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.31 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RK2
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![BU of 5rk2 by Molmil](/molmil-images/mine/5rk2) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z54633859 | Descriptor: | 2-[methyl(pyridin-2-yl)amino]ethan-1-ol, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.235 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKK
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![BU of 5rkk by Molmil](/molmil-images/mine/5rkk) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z275181224 | Descriptor: | N-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.43 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJO
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![BU of 5rjo by Molmil](/molmil-images/mine/5rjo) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00023827 | Descriptor: | 6-bromo-1,3-dihydro-2H-indol-2-one, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.22 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RK1
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![BU of 5rk1 by Molmil](/molmil-images/mine/5rk1) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1507502062 | Descriptor: | 6-methoxy-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.271 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKI
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![BU of 5rki by Molmil](/molmil-images/mine/5rki) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z198194396 | Descriptor: | 4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.268 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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8RU1
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![BU of 8ru1 by Molmil](/molmil-images/mine/8ru1) | Chromatin remodeling regulator CECR2 with in crystallo disulfide bond | Descriptor: | Chromatin remodeling regulator CECR2, GLYCEROL, SODIUM ION | Authors: | Fairhead, M, Strain-Damerell, C, Ye, M, Mackinnon, S.R, Pinkas, D, MacLean, E.M, Koekemoer, L, Damerell, D, Krojer, T, Arrowsmith, C.H, Edwards, A, Bountra, C, Yue, W, Burgess-Brown, N, Marsden, B, von Delft, F, Structural Genomics Consortium (SGC) | Deposit date: | 2024-01-29 | Release date: | 2024-03-06 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (1.66 Å) | Cite: | A fast, parallel method for efficiently exploring crystallization behaviour of large numbers of protein variants To Be Published
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8RU5
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![BU of 8ru5 by Molmil](/molmil-images/mine/8ru5) | ATPase family AAA domain containing 2 with crystallization epitope mutations V1022R:Q1027E | Descriptor: | 1,2-ETHANEDIOL, ATPase family AAA domain-containing protein 2 | Authors: | Fairhead, M, Strain-Damerell, C, Ye, M, Mackinnon, S.R, Pinkas, D, MacLean, E.M, Koekemoer, L, Damerell, D, Krojer, T, Arrowsmith, C.H, Edwards, A, Bountra, C, Yue, W, Burgess-Brown, N, Marsden, B, von Delft, F, Structural Genomics Consortium (SGC) | Deposit date: | 2024-01-30 | Release date: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.36 Å) | Cite: | A fast, parallel method for efficiently exploring crystallization behaviour of large numbers of protein variants To Be Published
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