5SC7
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![BU of 5sc7 by Molmil](/molmil-images/mine/5sc7) | CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with POB0120 | Descriptor: | (2R)-1',4'-dihydro-2'H-spiro[pyrrolidine-2,3'-quinolin]-2'-one, 1,2-ETHANEDIOL, CD44 antigen, ... | Authors: | Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O. | Deposit date: | 2021-09-14 | Release date: | 2021-09-22 | Method: | X-RAY DIFFRACTION (1.197 Å) | Cite: | CD44 PanDDA analysis group deposition To Be Published
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8CIU
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![BU of 8ciu by Molmil](/molmil-images/mine/8ciu) | The FERM domain of human moesin mutant H288A | Descriptor: | Moesin | Authors: | Bradshaw, W.J, Katis, V.L, Koekemoer, L, Bountra, C, von Delft, F, Brennan, P.E. | Deposit date: | 2023-02-10 | Release date: | 2023-03-01 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (2.393 Å) | Cite: | Discovery of FERM domain protein-protein interaction inhibitors for MSN and CD44 as a potential therapeutic approach for Alzheimer's disease. J.Biol.Chem., 299, 2023
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8CIT
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![BU of 8cit by Molmil](/molmil-images/mine/8cit) | The FERM domain of human moesin mutant L281R | Descriptor: | Moesin | Authors: | Bradshaw, W.J, Katis, V.L, Koekemoer, L, Bountra, C, von Delft, F, Brennan, P.E. | Deposit date: | 2023-02-10 | Release date: | 2023-03-01 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (2.536 Å) | Cite: | Discovery of FERM domain protein-protein interaction inhibitors for MSN and CD44 as a potential therapeutic approach for Alzheimer's disease. J.Biol.Chem., 299, 2023
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5RJP
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![BU of 5rjp by Molmil](/molmil-images/mine/5rjp) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024672 | Descriptor: | 4-bromo-1-(2-hydroxyethyl)pyridin-2(1H)-one, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.242 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RK3
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![BU of 5rk3 by Molmil](/molmil-images/mine/5rk3) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1501469697 | Descriptor: | 3-amino-1,6-dimethylpyridin-2(1H)-one, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.31 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKN
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![BU of 5rkn by Molmil](/molmil-images/mine/5rkn) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z373768900 | Descriptor: | N-(1-ethyl-1H-pyrazol-4-yl)cyclobutanecarboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.23 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJW
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![BU of 5rjw by Molmil](/molmil-images/mine/5rjw) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z256709556 | Descriptor: | 3-methylthiophene-2-carboxylic acid, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.514 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKB
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![BU of 5rkb by Molmil](/molmil-images/mine/5rkb) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z2004563941 | Descriptor: | (1S)-1-(1-cyclopentyl-1H-pyrazol-4-yl)ethan-1-ol, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.279 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKR
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![BU of 5rkr by Molmil](/molmil-images/mine/5rkr) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1432018343 | Descriptor: | (2S)-2-[(5-chloro-3-fluoropyridin-2-yl)amino]propan-1-ol, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.37 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJI
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![BU of 5rji by Molmil](/molmil-images/mine/5rji) | PanDDA analysis group deposition of ground-state model of PHIP | Descriptor: | PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.24 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJX
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![BU of 5rjx by Molmil](/molmil-images/mine/5rjx) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z285782452 | Descriptor: | N-methyl-2-(methylsulfonyl)aniline, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.291 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKD
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![BU of 5rkd by Molmil](/molmil-images/mine/5rkd) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z2168282707 | Descriptor: | (6S)-1-methyl-4,5,6,7-tetrahydro-1H-benzotriazole-6-carboxylic acid, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.237 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKU
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![BU of 5rku by Molmil](/molmil-images/mine/5rku) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z32367954 | Descriptor: | PH-interacting protein, ~{N}-cyclopropyl-1,3-benzodioxole-5-carboxamide | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.4 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJJ
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![BU of 5rjj by Molmil](/molmil-images/mine/5rjj) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00023833 | Descriptor: | 4-bromanyl-1,8-naphthyridine, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Method: | X-RAY DIFFRACTION (1.151 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJY
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![BU of 5rjy by Molmil](/molmil-images/mine/5rjy) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z383325512 | Descriptor: | N-[(1H-pyrazol-4-yl)methyl]acetamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.25 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKE
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![BU of 5rke by Molmil](/molmil-images/mine/5rke) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z906021418 | Descriptor: | 5-chloro-2-(propan-2-yl)pyrimidine-4-carboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.291 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKS
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![BU of 5rks by Molmil](/molmil-images/mine/5rks) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1696844792 | Descriptor: | 1-(diphenylmethyl)azetidin-3-ol, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.24 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJK
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![BU of 5rjk by Molmil](/molmil-images/mine/5rjk) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024661 | Descriptor: | 5-bromo-2-hydroxybenzonitrile, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.21 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RK0
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![BU of 5rk0 by Molmil](/molmil-images/mine/5rk0) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z30932204 | Descriptor: | N-[(4-sulfamoylphenyl)methyl]acetamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.24 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKG
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![BU of 5rkg by Molmil](/molmil-images/mine/5rkg) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1124201124 | Descriptor: | PH-interacting protein, ethyl 1~{H}-pyrazole-4-carboxylate | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.282 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKW
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![BU of 5rkw by Molmil](/molmil-images/mine/5rkw) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z27678561 | Descriptor: | N-(6-methoxy-1,3-benzothiazol-2-yl)cyclopropanecarboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.242 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RJU
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![BU of 5rju by Molmil](/molmil-images/mine/5rju) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z57261895 | Descriptor: | 2-cyclohexyl-N-(4H-1,2,4-triazol-4-yl)acetamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.32 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKA
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![BU of 5rka by Molmil](/molmil-images/mine/5rka) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z126932614 | Descriptor: | 2-[(methylsulfonyl)methyl]-1H-benzimidazole, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.33 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKO
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![BU of 5rko by Molmil](/molmil-images/mine/5rko) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z30620520 | Descriptor: | PH-interacting protein, cyclopropyl-[4-(4-fluorophenyl)piperazin-1-yl]methanone | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.42 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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5RKY
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![BU of 5rky by Molmil](/molmil-images/mine/5rky) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1796014543 | Descriptor: | 1-[(2-fluorophenyl)methyl]-N-methylcyclopropane-1-carboxamide, PH-interacting protein | Authors: | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | Deposit date: | 2020-06-02 | Release date: | 2020-06-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.38 Å) | Cite: | PanDDA analysis group deposition of ground-state model To Be Published
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