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PDB: 1 件

6Q8P
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Structure of CLK1 with bound N-methyl-10-nitropyrido[3,4-g]quinazolin-2-amine
分子名称: Dual specificity protein kinase CLK1, POTASSIUM ION, ~{N}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amine
著者Joerger, A.C, Chatterjee, D, Schroeder, M, Tazarki, H, Zeinyeh, W, Esvan, Y.J, Khiari, J, Josselin, B, Baratte, B, Bach, S, Ruchaud, S, Anizon, F, Giraud, F, Moreau, P, Knapp, S, Structural Genomics Consortium (SGC)
登録日2018-12-15
公開日2019-02-20
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis.
Eur J Med Chem, 166, 2019

222036

件を2024-07-03に公開中

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