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PDB: 1 件

4L6Q
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ROCK2 in complex with benzoxaborole
分子名称: 6-[4-(aminomethyl)-2-fluorophenoxy]-2,1-benzoxaborol-1(3H)-ol, Rho-associated protein kinase 2
著者Rock, F, Jarnagin, K.
登録日2013-06-12
公開日2013-10-02
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.79 Å)
主引用文献Linking phenotype to kinase: identification of a novel benzoxaborole hinge-binding motif for kinase inhibition and development of high-potency rho kinase inhibitors.
J.Pharmacol.Exp.Ther., 347, 2013

221051

件を2024-06-12に公開中

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