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PDB: 112 件

5U59
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BU of 5u59 by Molmil
Coiled Coil Peptide Metal Coordination Framework: Dimer Fold Grown with Citrate
分子名称: CITRIC ACID, COPPER (II) ION, Designed dimeric coiled coil peptide with two terpyridine side chains
著者Tavenor, N.A, Murnin, M.J, Horne, W.S.
登録日2016-12-06
公開日2017-02-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Supramolecular Metal-Coordination Polymers, Nets, and Frameworks from Synthetic Coiled-Coil Peptides.
J. Am. Chem. Soc., 139, 2017
6D07
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BU of 6d07 by Molmil
Crystal structure of the complex between human chromobox homolog 1 (CBX1) and H3K9me3 peptide
分子名称: Chromobox protein homolog 1, GLYCEROL, Histone H3.1
著者Arora, S, Horne, W.S, Islam, K.
登録日2018-04-10
公開日2019-04-10
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Engineering Methyllysine Writers and Readers for Allele-Specific Regulation of Protein-Protein Interactions.
J.Am.Chem.Soc., 141, 2019
5U5B
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BU of 5u5b by Molmil
Coiled Coil Peptide Metal Coordination Framework: Trimer Fold
分子名称: COPPER (II) ION, Designed trimeric coiled coil peptide with two terpyridine side chains, GLYCEROL
著者Tavenor, N.A, Murnin, M.J, Horne, W.S.
登録日2016-12-06
公開日2017-02-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Supramolecular Metal-Coordination Polymers, Nets, and Frameworks from Synthetic Coiled-Coil Peptides.
J. Am. Chem. Soc., 139, 2017
5US3
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Heterogeneous-backbone Foldamer Mimic of the Sp1-3 Zinc Finger
分子名称: Heterogeneous-Backbone Variant of the Sp1-3 Zinc Finger: N-Me-Ala3, N-Me-Arg10, beta-3-Asp15, ...
著者George, K.L, Horne, W.S.
登録日2017-02-13
公開日2017-05-31
最終更新日2024-07-10
実験手法SOLUTION NMR
主引用文献Heterogeneous-Backbone Foldamer Mimics of Zinc Finger Tertiary Structure.
J. Am. Chem. Soc., 139, 2017
4HU5
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Oxime side-chain cross-links in the GCN4-p1 dimeric coiled coil: Linear precursor
分子名称: ACETATE ION, GLYCEROL, General control protein GCN4
著者Haney, C.M, Horne, W.S.
登録日2012-11-02
公開日2013-08-21
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Oxime Side-Chain Cross-Links in an alpha-Helical Coiled-Coil Protein: Structure, Thermodynamics, and Folding-Templated Synthesis of Bicyclic Species.
Chemistry, 19, 2013
4KGS
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BU of 4kgs by Molmil
Backbone Modifications in the Protein GB1 Loops: beta-3-Val21, beta-3-Asp40
分子名称: GLYCEROL, Streptococcal Protein GB1 Backbone Modified Variant: beta-3-Val21, beta-3-Asp40
著者Reinert, Z.E, Lengyel, G.A, Horne, W.S.
登録日2013-04-29
公開日2013-09-04
最終更新日2024-07-10
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Protein-like Tertiary Folding Behavior from Heterogeneous Backbones.
J.Am.Chem.Soc., 135, 2013
4KGR
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BU of 4kgr by Molmil
Backbone Modifications in the Protein GB1 Helix: beta-3-Ala24, beta-3-Lys28, beta-3-Lys31, beta-3-Asn35
分子名称: GLYCEROL, Streptococcal Protein GB1 Backbone Modified Variant: beta-3-Ala24, beta-3-Lys28, ...
著者Reinert, Z.E, Lengyel, G.A, Horne, W.S.
登録日2013-04-29
公開日2013-09-04
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Protein-like Tertiary Folding Behavior from Heterogeneous Backbones.
J.Am.Chem.Soc., 135, 2013
4HU6
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BU of 4hu6 by Molmil
Oxime side-chain cross-links in the GCN4-p1 dimeric coiled coil: Cyclic product
分子名称: ACETATE ION, GLYCEROL, General control protein GCN4
著者Haney, C.M, Horne, W.S.
登録日2012-11-02
公開日2013-08-21
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Oxime Side-Chain Cross-Links in an alpha-Helical Coiled-Coil Protein: Structure, Thermodynamics, and Folding-Templated Synthesis of Bicyclic Species.
Chemistry, 19, 2013
4KGT
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BU of 4kgt by Molmil
Backbone Modifications in the Protein GB1 Turns: Aib10, D-Pro47
分子名称: Streptococcal Protein GB1 Backbone Modified Variant: Aib10, D-Pro47
著者Reinert, Z.E, Lengyel, G.A, Horne, W.S.
登録日2013-04-29
公開日2013-09-04
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Protein-like Tertiary Folding Behavior from Heterogeneous Backbones.
J.Am.Chem.Soc., 135, 2013
3F87
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An alpha/beta-Peptide Helix Bundle with a Pure beta-Amino Acid Core and a Distinctive Quarternary Structure: GCN4pLI derivative with beta residues at a and d heptad positions - higher symmetry crystal
分子名称: GCN4pLI-betaAD, IODIDE ION
著者Giuliano, M.W, Horne, W.S, Gellman, S.H.
登録日2008-11-11
公開日2009-07-21
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献An alpha/beta-peptide helix bundle with a pure beta3-amino acid core and a distinctive quaternary structure.
J.Am.Chem.Soc., 131, 2009
3F86
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An alpha/beta-Peptide Helix Bundle with a Pure beta-Amino Acid Core and a Distinctive Quaternary Structure: GCN4pLI derivative with beta residues at a and d heptad positions
分子名称: GCN4pLI-betaAD
著者Giuliano, M.W, Horne, W.S, Gellman, S.H.
登録日2008-11-11
公開日2009-07-21
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献An alpha/beta-peptide helix bundle with a pure beta3-amino acid core and a distinctive quaternary structure.
J.Am.Chem.Soc., 131, 2009
3UE8
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BU of 3ue8 by Molmil
Kynurenine Aminotransferase II Inhibitors
分子名称: (5-hydroxy-4-{[(1-hydroxy-2-oxo-1,2-dihydroquinolin-3-yl)amino]methyl}-6-methylpyridin-3-yl)methyl dihydrogen phosphate, CHLORIDE ION, Kynurenine/alpha-aminoadipate aminotransferase, ...
著者Dounay, A.B, Anderson, M, Bechle, B.M, Campbell, B.M, Claffey, M.M, Evdokimov, A, Edelweiss, E, Fonseca, K.R, Gan, X, Ghosh, S, Hayward, M.M, Horner, W, Kim, J.Y, McAllister, L.A, Pandit, J, Paradis, V, Parikh, V.D, Reese, M.R, Rong, S.B, Salafia, M.A, Schuyten, K, Strick, C.A, Tuttle, J.B, Valentine, J, Wang, H, Zawadzke, L.E, Verhoest, P.R.
登録日2011-10-28
公開日2012-02-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.22 Å)
主引用文献Discovery of Brain-Penetrant, Irreversible Kynurenine Aminotransferase II Inhibitors for Schizophrenia.
ACS Med Chem Lett, 3, 2012

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件を2024-07-17に公開中

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