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PDB: 6 results

1T4E
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BU of 1t4e by Molmil
Structure of Human MDM2 in complex with a Benzodiazepine Inhibitor
Descriptor: (4-CHLOROPHENYL)[3-(4-CHLOROPHENYL)-7-IODO-2,5-DIOXO-1,2,3,5-TETRAHYDRO-4H-1,4-BENZODIAZEPIN-4-YL]ACETIC ACID, Ubiquitin-protein ligase E3 Mdm2
Authors:Grasberger, B.L, Schubert, C, Koblish, H.K, Carver, T.E, Franks, C.F, Zhao, S.Y, Lu, T, LaFrance, L.V, Parks, D.J.
Deposit date:2004-04-29
Release date:2005-02-08
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Discovery and cocrystal structure of benzodiazepinedione HDM2 antagonists that activate p53 in cells
J.Med.Chem., 48, 2005
1T4F
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BU of 1t4f by Molmil
Structure of human MDM2 in complex with an optimized p53 peptide
Descriptor: SULFATE ION, Ubiquitin-protein ligase E3 Mdm2, optimized p53 peptide
Authors:Grasberger, B.L, Schubert, C, Koblish, H.K, Carver, T.E, Franks, C.F, Zhao, S.Y, Lu, T, LaFrance, L.V, Parks, D.J.
Deposit date:2004-04-29
Release date:2005-02-08
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Discovery and cocrystal structure of benzodiazepinedione HDM2 antagonists that activate p53 in cells
J.Med.Chem., 48, 2005
1ATB
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BU of 1atb by Molmil
HIGH-RESOLUTION STRUCTURE OF ASCARIS TRYPSIN INHIBITOR IN SOLUTION: DIRECT EVIDENCE FOR A PH INDUCED CONFORMATIONAL TRANSITION IN THE REACTIVE SITE
Descriptor: ASCARIS TRYPSIN INHIBITOR
Authors:Clore, G.M, Grasberger, B.L, Gronenborn, A.M.
Deposit date:1994-05-20
Release date:1994-08-31
Last modified:2022-02-16
Method:SOLUTION NMR
Cite:High-resolution structure of Ascaris trypsin inhibitor in solution: direct evidence for a pH-induced conformational transition in the reactive site.
Structure, 2, 1994
1ATD
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BU of 1atd by Molmil
HIGH-RESOLUTION STRUCTURE OF ASCARIS TRYPSIN INHIBITOR IN SOLUTION: DIRECT EVIDENCE FOR A PH INDUCED CONFORMATIONAL TRANSITION IN THE REACTIVE SITE
Descriptor: ASCARIS TRYPSIN INHIBITOR
Authors:Clore, G.M, Grasberger, B.L, Gronenborn, A.M.
Deposit date:1994-05-20
Release date:1994-08-31
Last modified:2022-02-16
Method:SOLUTION NMR
Cite:High-resolution structure of Ascaris trypsin inhibitor in solution: direct evidence for a pH-induced conformational transition in the reactive site.
Structure, 2, 1994
1ATE
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BU of 1ate by Molmil
HIGH-RESOLUTION STRUCTURE OF ASCARIS TRYPSIN INHIBITOR IN SOLUTION: DIRECT EVIDENCE FOR A PH INDUCED CONFORMATIONAL TRANSITION IN THE REACTIVE SITE
Descriptor: ASCARIS TRYPSIN INHIBITOR
Authors:Clore, G.M, Grasberger, B.L, Gronenborn, A.M.
Deposit date:1994-05-20
Release date:1994-08-31
Last modified:2022-02-16
Method:SOLUTION NMR
Cite:High-resolution structure of Ascaris trypsin inhibitor in solution: direct evidence for a pH-induced conformational transition in the reactive site.
Structure, 2, 1994
1ATA
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BU of 1ata by Molmil
HIGH-RESOLUTION STRUCTURE OF ASCARIS TRYPSIN INHIBITOR IN SOLUTION: DIRECT EVIDENCE FOR A PH INDUCED CONFORMATIONAL TRANSITION IN THE REACTIVE SITE
Descriptor: ASCARIS TRYPSIN INHIBITOR
Authors:Clore, G.M, Grasberger, B.L, Gronenborn, A.M.
Deposit date:1994-05-20
Release date:1994-08-31
Last modified:2022-02-16
Method:SOLUTION NMR
Cite:High-resolution structure of Ascaris trypsin inhibitor in solution: direct evidence for a pH-induced conformational transition in the reactive site.
Structure, 2, 1994

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