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PDB: 1 件

4JVG
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B-Raf Kinase in Complex with Birb796
分子名称: 1-(5-TERT-BUTYL-2-P-TOLYL-2H-PYRAZOL-3-YL)-3-[4-(2-MORPHOLIN-4-YL-ETHOXY)-NAPHTHALEN-1-YL]-UREA, Serine/threonine-protein kinase B-raf
著者Lavoie, H, Thevakumaran, N, Gavory, G, Li, J, Padeganeh, A, Guiral, S, Duchaine, J, Mao, D.Y.L, Bouvier, M, Sicheri, F, Therrien, M.
登録日2013-03-25
公開日2013-05-29
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.09 Å)
主引用文献Inhibitors that stabilize a closed RAF kinase domain conformation induce dimerization.
Nat.Chem.Biol., 9, 2013

221051

件を2024-06-12に公開中

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