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PDB: 1 件

5CLM
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1,4-Oxazine BACE1 inhibitors
分子名称: Beta-secretase 1, CHLORIDE ION, IODIDE ION, ...
著者Rombouts, F, Tresadern, G, Delgado, O, Martinez Lamenca, C, Van Gool, M, Garcia-Molina, A, Alonso De Diego, S, Oehlrich, D, Prokopcova, H, Alonso, J.M, Austin, N, Borghys, H, Van Brandt, S, Surkyn, M, De Cleyn, M, Vos, A, Alexander, R, MacDonald, G, Moechars, D, Trabanco, A, Gijsen, H.
登録日2015-07-16
公開日2015-09-30
最終更新日2015-11-04
実験手法X-RAY DIFFRACTION (2.61 Å)
主引用文献1,4-Oxazine beta-Secretase 1 (BACE1) Inhibitors: From Hit Generation to Orally Bioavailable Brain Penetrant Leads.
J.Med.Chem., 58, 2015

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件を2024-07-17に公開中

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