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PDB: 1 件

8RQ9
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BU of 8rq9 by Molmil
Crystal structure of PROTAC CFT-1297 in complex with CRBN-midi and BRD4(BD2)
分子名称: (3~{S})-3-[7-[1-[7-[4-[6-(4-chlorophenyl)-1-methyl-spiro[[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4,1'-cyclopropane]-8-yl]pyrazol-1-yl]heptyl]piperidin-4-yl]-3-oxidanylidene-1~{H}-isoindol-2-yl]piperidine-2,6-dione, Bromodomain-containing protein 4, Protein cereblon, ...
著者Darren, D, Ramachandran, S, Kroupova, A, Zollman, D, Ciulli, A.
登録日2024-01-17
公開日2024-09-25
実験手法X-RAY DIFFRACTION (2.91 Å)
主引用文献Design of a Cereblon construct for crystallographic and biophysical studies of protein degraders
To Be Published

225399

件を2024-09-25に公開中

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