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PDB: 1 件

4M7B
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Human tankyrase 2 - catalytic Parp domain in complex with an inhibitor UPF1854
分子名称: 4-{2-[(6-methyl[1,2,4]triazolo[4,3-b]pyridazin-8-yl)amino]ethyl}phenol, SULFATE ION, Tankyrase-2, ...
著者Karlberg, T, Camaioni, E, Schuler, H.
登録日2013-08-12
公開日2014-03-12
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Design, Synthesis, Crystallographic Studies, and Preliminary Biological Appraisal of New Substituted Triazolo[4,3-b]pyridazin-8-amine Derivatives as Tankyrase Inhibitors.
J.Med.Chem., 57, 2014

219869

件を2024-05-15に公開中

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