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PDB: 4 件

4HEJ
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BU of 4hej by Molmil
Discovery of Selective and Potent Inhibitors of Gram-positive Bacterial Thymidylate Kinase (TMK): Compund 16
分子名称: 5-methyl-1-[(3S)-1-{3-[3-(trifluoromethyl)phenoxy]benzyl}piperidin-3-yl]pyrimidine-2,4(1H,3H)-dione, Thymidylate kinase
著者Martinez-Botella, G, Breen, J, Duffy, J, Dumas, J, Geng, B, Gowers, I, Green, O, Guler, S, Hentemann, M, Hernandez-Juan, F, Joseph-McCarthy, D, Kawatkar, S, Larsen, N, Lazari, O, Loch, J, Macritchie, J.
登録日2012-10-03
公開日2012-10-24
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Discovery of Selective and Potent Inhibitors of Gram-Positive Bacterial Thymidylate Kinase (TMK).
J.Med.Chem., 55, 2012
4Y0A
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BU of 4y0a by Molmil
Shikimate kinase from Acinetobacter baumannii in complex with shikimate
分子名称: (3R,4S,5R)-3,4,5-TRIHYDROXYCYCLOHEX-1-ENE-1-CARBOXYLIC ACID, SULFATE ION, Shikimate kinase
著者Sutton, K.A, Breen, J, MacDonald, U, Beanan, J.M, Olson, R, Russo, T.A, Schultz, L.W, Umland, T.C.
登録日2015-02-05
公開日2015-08-12
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.911 Å)
主引用文献Structure of shikimate kinase, an in vivo essential metabolic enzyme in the nosocomial pathogen Acinetobacter baumannii, in complex with shikimate.
Acta Crystallogr.,Sect.D, 71, 2015
5BUF
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2.37 Angstrom Structure of EPSP Synthase from acinetobacter baumannii
分子名称: 3-phosphoshikimate 1-carboxyvinyltransferase, CHLORIDE ION
著者Sutton, K.A, Schultz, L.W, Breen, J, Graham, J, Umland, T.C.
登録日2015-06-03
公開日2016-02-17
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.37 Å)
主引用文献Crystal structure of 5-enolpyruvylshikimate-3-phosphate (EPSP) synthase from the ESKAPE pathogen Acinetobacter baumannii.
Acta Crystallogr.,Sect.F, 72, 2016
5BS5
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EPSP synthase from Acinetobacter baumannii
分子名称: 3-phosphoshikimate 1-carboxyvinyltransferase
著者Sutton, K.A, Schultz, L.W, Russo, T.A, Breen, J, Umland, T.C.
登録日2015-06-01
公開日2016-02-24
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献EPSP synthase from Acinetobacter baumannii
Acta Crystallogr.,Sect.F, 2016

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件を2024-05-22に公開中

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