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PDB: 3 件

4LP0
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BU of 4lp0 by Molmil
Crystal structure of a topoisomerase ATP inhibitor
分子名称: 6'-[(ethylcarbamoyl)amino]-4'-[4-(trifluoromethyl)-1,3-thiazol-2-yl]-3,3'-bipyridine-5-carboxylic acid, Topoisomerase IV subunit B
著者Basarab, G.S, Manchester, J.I, Bist, S, Boriack-Sjodin, P.A, Dangel, B, Illingsworth, R, Uria-Nickelsen, M, Sherer, B.A, Sriram, S, Eakin, A.E.
登録日2013-07-14
公開日2013-11-13
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Fragment-to-Hit-to-Lead Discovery of a Novel Pyridylurea Scaffold of ATP Competitive Dual Targeting Type II Topoisomerase Inhibiting Antibacterial Agents.
J.Med.Chem., 56, 2013
8P33
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BU of 8p33 by Molmil
BB0238 from Borrelia burgdorferi
分子名称: BB0238
著者Brangulis, K, Foor, S.D, Shakya, A.K, Rana, V.S, Bista, S, Kitsou, C, Ronzetti, M, Linden, S.B, Altieri, A.S, Akopjana, I, Baljinnyam, B, Nelson, D.C, Simeonov, A, Herzberg, O, Caimano, M.J, Pal, U.
登録日2023-05-16
公開日2023-10-11
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献A unique borrelial protein facilitates microbial immune evasion.
Mbio, 14, 2023
8P32
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BU of 8p32 by Molmil
BB0238 from Borrelia burgdorferi, Se-Met data for Leu240Met mutant
分子名称: BB0238
著者Brangulis, K, Foor, S.D, Shakya, A.K, Rana, V.S, Bista, S, Kitsou, C, Ronzetti, M, Linden, S.B, Altieri, A.S, Akopjana, I, Baljinnyam, B, Nelson, D.C, Simeonov, A, Herzberg, O, Caimano, M.J, Pal, U.
登録日2023-05-16
公開日2023-10-11
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献A unique borrelial protein facilitates microbial immune evasion.
Mbio, 14, 2023

223166

件を2024-07-31に公開中

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